SCHEMBL9025564

SCHEMBL9025564

O=c1[nH]c(=O)n([C@@H]2[C@@H](F)[C@H](CO)[C@H]2CO)cc1I

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TK1 P04183 4/20 0.50
PYGM P11217 1/20 0.49
P2RY6 Q15077 2/20 0.36
P2RY14 Q15391 2/20 0.36
BLM P54132 2/20 0.36
CYP1A2 P05177 1/20 0.36
GRIA1 P42261 1/20 0.36
GRIA2 P42262 1/20 0.36
GRIA4 P48058 1/20 0.36
KMT2A Q03164 1/20 0.36
GRIK5 Q16478 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TK2 O00142 2/20 0.35
LMNA P02545 2/20 0.35
ALDH1A1 P00352 1/20 0.35
ALB P02768 1/20 0.35
POLB P06746 1/20 0.35
ADRA1A P35348 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
TYMP P19971 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025572 1.00 TK1 (0.50) TK1PYGMP2RY6P2RY14BLM
SCHEMBL9310440 0.90 TK1 (0.56) TK1PYGMP2RY6P2RY14BLM
SCHEMBL10827402 0.88 PYGM (0.52) TK1PYGMP2RY6P2RY14TK2
SCHEMBL10827761 0.88 PYGM (0.52) TK1PYGMP2RY6P2RY14TK2
SCHEMBL10827403 0.88 PYGM (0.52) TK1PYGMP2RY6P2RY14TK2
SCHEMBL10827758 0.88 PYGM (0.52) TK1PYGMP2RY6P2RY14TK2
SCHEMBL10827405 0.88 PYGM (0.52) TK1PYGMP2RY6P2RY14TK2
SCHEMBL9024558 0.83 LMNA (0.52) TK1BLMLMNAALDH1A1ALB
SCHEMBL9025958 0.83 LMNA (0.52) TK1BLMLMNAALDH1A1ALB
SCHEMBL9025283 0.81 TK2 (0.45) TK1BLMCYP1A2TK2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458363-B1 Fluorinated bis(hydroxymethyl) cyclobutyl purines and pyrimidines SQUIBB & SONS INC (US) 1996-02-07 EP claimed
WO-1991018969-A1 FLUORINATED BIS(HYDROXYMETHYL)CYCLOBUTYL PURINES AND PYRIMIDINES E.R. SQUIBB & SONS, INC. (US) 1991-12-12 WO claimed
EP-0458363-A1 Fluorinated bis(hydroxymethyl) cyclobutyl purines and pyrimidines E.R. SQUIBB & SONS, INC. (US) 1991-11-27 EP claimed
EP-0458363-B1 Fluorinated bis(hydroxymethyl) cyclobutyl purines and pyrimidines SQUIBB & SONS INC (US) 1996-02-07 EP disclosed
WO-1991018969-A1 FLUORINATED BIS(HYDROXYMETHYL)CYCLOBUTYL PURINES AND PYRIMIDINES E.R. SQUIBB & SONS, INC. (US) 1991-12-12 WO disclosed
EP-0458363-A1 Fluorinated bis(hydroxymethyl) cyclobutyl purines and pyrimidines E.R. SQUIBB & SONS, INC. (US) 1991-11-27 EP disclosed