SCHEMBL902859

SCHEMBL902859

Cc1cnc(-c2nc3ccc(Cl)cc3[nH]2)cn1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.63
METAP2 P50579 2/20 0.58
METAP1 P53582 2/20 0.58
CBFB Q13951 1/20 0.58
ALDH1A1 P00352 2/20 0.56
HPGD P15428 2/20 0.56
KDM4E B2RXH2 1/20 0.56
MEN1 O00255 1/20 0.56
TP53 P04637 1/20 0.56
CYP3A4 P08684 1/20 0.56
MAPT P10636 1/20 0.56
MAPK1 P28482 1/20 0.56
KMT2A Q03164 1/20 0.56
HSD17B10 Q99714 1/20 0.56
FTO Q9C0B1 1/20 0.56
NPC1 O15118 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.50
P2RY6 Q15077 1/20 0.49
DGAT1 O75907 5/20 0.47
AMY1A P0DUB6 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13286844 0.81 NPC1 (0.57) ADORA3METAP2METAP1CBFBALDH1A1
SCHEMBL903006 0.80 METAP2 (0.61) METAP2METAP1CBFBNPC1DGAT1
SCHEMBL902815 0.79 CBFB (0.64) CBFBDGAT1
SCHEMBL34849 0.78 ADORA3 (0.47) ADORA3METAP2METAP1CBFBALDH1A1
SCHEMBL902354 0.77 CBFB (0.64) CBFBNPC1P2RY6DGAT1BACE1
SCHEMBL4900779 0.77 METAP2 (0.57) ADORA3METAP2METAP1CBFBALDH1A1
SCHEMBL34855 0.77 NPC1 (0.55) ADORA3METAP2METAP1CBFBALDH1A1
SCHEMBL5952973 0.77 METAP2 (0.57) ADORA3METAP2METAP1CBFBALDH1A1
SCHEMBL29898236 0.72 KDM4E (1.00) ADORA3METAP2METAP1CBFBALDH1A1
SCHEMBL8337597 0.72 KDM4E (1.00) ADORA3METAP2METAP1CBFBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed