SCHEMBL9033216

SCHEMBL9033216

O=C(O)NC(Cc1ccccc1)C(O)c1ccc(CN2CCCC2)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 2/20 0.38
FAAH O00519 1/20 0.38
HRH3 Q9Y5N1 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ACACB O00763 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8703407 0.86 HRH3 (0.39) ALDH1A1CYP2D6CYP2C9CYP3A4CYP2C19
SCHEMBL8698602 0.81 HRH3 (0.38) ALDH1A1HRH3KDM4EMAPTHTT
SCHEMBL8702811 0.80 HRH3 (0.40) ALDH1A1CYP2D6CYP2C9CYP3A4CYP2C19
SCHEMBL9032268 0.80 HRH3 (0.46) ALDH1A1SMN1; SMN2GAAHRH3KDM4E
SCHEMBL8697846 0.78 OPRK1 (0.44) CYP3A4SMN1; SMN2HRH3LMNATSHR
SCHEMBL9034272 0.75 ATM (0.45) ALDH1A1CYP3A4SMN1; SMN2HRH3LMNA
SCHEMBL9032737 0.75 CTSL (0.44) CYP2D6CYP2C9CYP3A4CYP2C19SMN1; SMN2
SCHEMBL8701081 0.74 SIGMAR1 (0.38) ALDH1A1SMN1; SMN2HRH3MEN1KMT2A
SCHEMBL9031818 0.74 CTSL (0.44) CYP2D6CYP2C9CYP3A4CYP2C19SMN1; SMN2
SCHEMBL9033877 0.74 SMN1; SMN2 (0.44) ALDH1A1CYP2D6CYP2C9SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1121713-A serine derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-05-01 CN disclosed
EP-0696586-A1 SERINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed