SCHEMBL9033992

SCHEMBL9033992

OC1(CCc2ccc3[nH]cc(C4=CCNCC4)c3c2)CCCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.53
KDM4E B2RXH2 4/20 0.52
ALDH1A1 P00352 4/20 0.52
HSD17B10 Q99714 4/20 0.52
HTR2C P28335 3/20 0.52
MAPT P10636 3/20 0.52
HTR1D P28221 3/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
CYP1A2 P05177 2/20 0.52
CYP3A4 P08684 2/20 0.52
MAPK1 P28482 1/20 0.52
BRCA1 P38398 1/20 0.52
DRD2 P14416 2/20 0.50
ALOX15 P16050 1/20 0.50
JAK2 O60674 1/20 0.46
PRKD3 O94806 1/20 0.46
MARK3 P27448 1/20 0.46
PRKCI P41743 1/20 0.46
PRKCD Q05655 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13533314 0.81 HTR6 (0.63) HTR6KDM4EALDH1A1HSD17B10HTR2C
SCHEMBL8914068 0.77 OPRM1 (0.65) KDM4EDRD2ALOX15HTR1AHTR2A
SCHEMBL3836149 0.74 HTR6 (0.67) HTR6KDM4EALDH1A1HSD17B10HTR2C
SCHEMBL8916861 0.73 NMT2 (0.48) HTR6HTR2CHTR1DCYP1A2CYP3A4
SCHEMBL1675799 0.71 HTR6 (0.67) HTR6KDM4EALDH1A1HSD17B10HTR2C
SCHEMBL2783986 0.71 HTR6 (0.67) HTR6KDM4EALDH1A1HSD17B10HTR2C
SCHEMBL7460028 0.71 HTR6 (0.67) HTR6KDM4EALDH1A1HSD17B10HTR2C
SCHEMBL2778860 0.71 HTR6 (0.67) HTR6KDM4EALDH1A1HSD17B10HTR2C
SCHEMBL6631651 0.71 KDM4E (0.70) HTR6KDM4EALDH1A1HSD17B10HTR2C
SCHEMBL8915519 0.71 NMT2 (0.42) HTR6HTR2CHTR1DCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0695301-B1 INDOLE DERIVATIVES AS 5-HT1-LIKE AGONISTS FOR USE IN MIGRAINE PFIZER LTD (GB) 1996-10-30 EP disclosed