SCHEMBL8915519

SCHEMBL8915519

OC1(CCc2ccc3[nH]cc(C4CCNC4)c3c2)CCCC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NMT2 O60551 1/20 0.42
NMT1 P30419 1/20 0.42
APP P05067 3/20 0.41
HTR2C P28335 2/20 0.40
ADRB2 P07550 1/20 0.40
HTR1D P28221 5/20 0.39
HTR1B P28222 5/20 0.39
HTR1A P08908 1/20 0.39
IDO1 P14902 1/20 0.37
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
CHEK1 O14757 1/20 0.36
WEE1 P30291 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
THPO P40225 1/20 0.35
HTR6 P50406 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916861 0.93 NMT2 (0.48) NMT2NMT1APPHTR2CADRB2
SCHEMBL8913781 0.82 HTR1D (0.59) APPHTR1DHTR1BHTR1ANOS3
SCHEMBL9033996 0.77 IDO1 (0.36) HTR1DHTR1BHTR1AIDO1
SCHEMBL27294918 0.76 NMT2 (0.48) NMT2NMT1APPHTR2CADRB2
SCHEMBL7665068 0.73 HTR6 (0.54) HTR2CHTR1DHTR1BHTR1AHTR6
SCHEMBL9033992 0.71 HTR6 (0.53) HTR2CHTR1DHTR1BHTR1ACYP1A2
SCHEMBL8913687 0.71 HTR6 (0.54) HTR2CHTR1DHTR1BHTR1AHTR6
SCHEMBL9040223 0.71 SLC6A4 (0.32) HTR1DHTR1BHTR6
SCHEMBL1445394 0.71 GABRP (0.54) APPHTR2CADRB2HTR1DHTR1B
SCHEMBL31328282 0.71 SLC6A4 (0.56) APPHTR2CADRB2HTR1AIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607960-A Indole derivatives as 5-HT1-like agonists for use in migraine PFIZER INC. (US) 1997-03-04 US disclosed
EP-0695301-B1 INDOLE DERIVATIVES AS 5-HT1-LIKE AGONISTS FOR USE IN MIGRAINE PFIZER LTD (GB) 1996-10-30 EP disclosed
WO-1994024127-A1 INDOLE DERIVATIVES AS 5-H1-LIKE AGONISTS FOR USE IN MIGRAINE PFIZER LIMITED (GB) 1994-10-27 WO disclosed