SCHEMBL9035328

SCHEMBL9035328

Brc1ccc(Br)nc1.O=C(O)c1ccc(Br)nc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
KDM4E B2RXH2 1/20 0.55
P4HA1 P13674 3/20 0.53
P4HTM Q9NXG6 2/20 0.53
MIF P14174 1/20 0.52
GABRP O00591 1/20 0.50
GABRD O14764 1/20 0.50
GABRA1 P14867 1/20 0.50
GABRB1 P18505 1/20 0.50
GABRG2 P18507 1/20 0.50
GABRB3 P28472 1/20 0.50
GABRA5 P31644 1/20 0.50
GABRA3 P34903 1/20 0.50
GABRA2 P47869 1/20 0.50
GABRB2 P47870 1/20 0.50
GABRA4 P48169 1/20 0.50
GABRE P78334 1/20 0.50
GABRA6 Q16445 1/20 0.50
GABRG1 Q8N1C3 1/20 0.50
GABRG3 Q99928 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38414 0.92 P4HA1 (0.61) ALDH1A1P4HA1P4HTMMIFGABRP
SCHEMBL29751460 0.92 P4HA1 (0.61) ALDH1A1P4HA1P4HTMMIFGABRP
Hydrochloric Acid SCHEMBL1871783 0.90 P4HA1 (0.59) ALDH1A1P4HA1P4HTMMIFGABRP
Nitrous Acid SCHEMBL27425985 0.85 P4HA1 (0.53) ALDH1A1P4HA1P4HTMMIFGABRP
SCHEMBL16841 0.78
SCHEMBL29411198 0.78
SCHEMBL5973043 0.77 RXFP1 (0.44) ALDH1A1P4HA1P4HTMMIFGABRP
Formaldehyde SCHEMBL27841183 0.77 ALDH1A1 (0.46) ALDH1A1KDM4ETSHR
SCHEMBL3500140 0.76 HCAR3 (0.69) HCAR3
SCHEMBL3500869 0.76 NPC1 (0.66) KDM4ECYP1A2CYP2C9CYP2C19HCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712397-A1 AMIDE DERIVATIVES AS 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-05-22 EP disclosed
WO-1995004729-A1 AMIDE DERIVATIVES AS 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-02-16 WO disclosed