SCHEMBL903534

SCHEMBL903534

COc1ccc(-c2[nH]c3ccc(OC)cc3c2F)c(O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.53
MEN1 O00255 5/20 0.53
KMT2A Q03164 5/20 0.53
ALDH1A1 P00352 5/20 0.53
KDM4E B2RXH2 5/20 0.53
HSD17B10 Q99714 3/20 0.53
MAPT P10636 3/20 0.53
GFER P55789 2/20 0.53
TSHR P16473 1/20 0.53
HPGD P15428 3/20 0.50
CDK1 P06493 2/20 0.47
CCNB1 P14635 2/20 0.47
GSK3B P49841 2/20 0.47
CCNB2 O95067 1/20 0.47
GSK3A P49840 1/20 0.47
CDK5 Q00535 1/20 0.47
CDK5R1 Q15078 1/20 0.47
CCNB3 Q8WWL7 1/20 0.47
APOBEC3A P31941 1/20 0.47
APOBEC3G Q9HC16 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL903542 0.91 ALOX5 (0.48) ALOX5MEN1KMT2AALDH1A1KDM4E
SCHEMBL27255944 0.79 ALOX5 (0.47) ALOX5MEN1KMT2AALDH1A1KDM4E
SCHEMBL22628563 0.76 CTSV (0.49) ALOX5MEN1KMT2AALDH1A1KDM4E
SCHEMBL31053079 0.76 CTSV (0.49) ALOX5MEN1KMT2AALDH1A1KDM4E
SCHEMBL17452876 0.74 ALDH1A1 (0.63) ALOX5MEN1KMT2AALDH1A1KDM4E
SCHEMBL903529 0.74 AR (0.50) ALOX5MEN1KMT2AALDH1A1KDM4E
SCHEMBL29233384 0.73 HSD17B10 (0.78) ALOX5MEN1KMT2AALDH1A1KDM4E
SCHEMBL10215057 0.71 KIF11 (0.37) MEN1KMT2AALDH1A1KDM4EHSD17B10
SCHEMBL2597652 0.71 ALDH1A1 (1.00) MEN1KMT2AALDH1A1KDM4EHSD17B10
SCHEMBL29391519 0.71 ALDH1A1 (1.00) MEN1KMT2AALDH1A1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041014-A1 TETRACYCLIC INDOLE DERIVATIVES FOR TREATING HEPATITIS C VIRUS INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed
WO-2012040923-A1 TETRACYCLIC INDOLE DERIVATIVES AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed