SCHEMBL9035904

SCHEMBL9035904

Clc1ccc2c(N3CCCCC3)noc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 2/20 0.48
HTR1A P08908 1/20 0.47
HTR2A P28223 1/20 0.47
CHKA P35790 1/20 0.46
MAPK13 O15264 1/20 0.43
PKM P14618 1/20 0.43
ALOX15 P16050 1/20 0.43
CASP1 P29466 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTR3A P46098 3/20 0.43
CHRNA7 P36544 2/20 0.43
GFER P55789 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9037461 0.98 MAT2A (0.47) MAT2AHTR1AHTR2ACHKAMAPK13
SCHEMBL1840383 0.85 HRH4 (0.48) HTR1AHTR2AHTR3ACHRNA7TP53
SCHEMBL30777987 0.81 HTR2A (0.48) HTR1AHTR2AHTR3ACHRNA7NPC1
SCHEMBL23064293 0.81 HTR2A (0.48) HTR1AHTR2AHTR3ACHRNA7NPC1
SCHEMBL13448295 0.81 HTT (0.54) HTR1AHTR2ANPC1TP53RAB9A
SCHEMBL531012 0.81 ACHE (0.52) HTR1AHTR2AMAPK13HTR3ACHRNA7
SCHEMBL5905921 0.81 MAPK13 (0.43) MAPK13ALOX15NPC1HPGDTSHR
Hydrochloric Acid SCHEMBL14128737 0.80 ACHE (0.51) HTR1AHTR2AMAPK13HTR3ACHRNA7
SCHEMBL14748231 0.79 HTR2A (0.51) HTR1AHTR2A
SCHEMBL23074485 0.78 MAPT (0.46) HTR1AHTR2AHSD17B10TP53HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0511610-B1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST ROUSSEL PHARMA (US) 1996-09-11 EP disclosed
US-5225412-A Antipsychotic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-06 US disclosed
EP-0511610-A1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-11-04 EP disclosed
US-5143923-A Psychological disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-09-01 US disclosed