SCHEMBL9036686

SCHEMBL9036686

OC1(c2ccccc2C(F)(F)F)CCC(N2CCNCC2)CC1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPV6 Q9H1D0 2/20 0.59
HPGD P15428 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTR2C P28335 4/20 0.40
HTR2A P28223 1/20 0.40
OPRM1 P35372 2/20 0.39
OPRD1 P41143 2/20 0.39
OPRL1 P41146 2/20 0.39
PDK2 Q15119 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
EPHX2 P34913 1/20 0.37
HTR6 P50406 1/20 0.37
KCNH2 Q12809 1/20 0.37
GRIN2B Q13224 1/20 0.37
HDAC4 P56524 1/20 0.36
TRPV5 Q9NQA5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964019 0.82 TRPV6 (0.53) TRPV6OPRM1OPRD1OPRL1PDK2
SCHEMBL1513500 0.80 SIGMAR1 (0.53) TRPV6HTR2COPRM1OPRD1OPRL1
SCHEMBL29980126 0.80 SIGMAR1 (0.53) TRPV6HTR2COPRM1OPRD1OPRL1
SCHEMBL8142385 0.80 TRPV6 (0.52) TRPV6OPRM1OPRD1OPRL1KDM4E
Hydrochloric Acid SCHEMBL3326791 0.79 SIGMAR1 (0.51) TRPV6HTR2COPRM1OPRD1OPRL1
SCHEMBL9036683 0.76 OPRL1 (0.45) TRPV6HTR2COPRM1OPRD1OPRL1
SCHEMBL7040982 0.76 TRPV6 (0.63) TRPV6OPRM1OPRD1OPRL1KDM4E
SCHEMBL11793878 0.76 TRPV6 (0.48) TRPV6HTR2COPRM1OPRD1OPRL1
SCHEMBL6964017 0.73 TRPV6 (0.41) TRPV6HTR2CPDK2HDAC4
SCHEMBL1919333 0.72 HDAC4 (0.57) TRPV6OPRM1OPRD1OPRL1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0546583-B1 Piperazinyl-and piperidinyl-cyclohexanols BRISTOL MYERS SQUIBB CO (US) 1996-05-22 EP disclosed
US-5478828-A Anxiolytic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-12-26 US disclosed
US-5387593-A Anxiolytic agents BRISTON-MYERS SQUIBB (US) 1995-02-07 US disclosed
EP-0546583-A1 Piperazinyl-and piperidinyl-cyclohexanols Bristol-Myers Squibb Company (US) 1993-06-16 EP disclosed