SCHEMBL9037155

SCHEMBL9037155

COc1cccc2c1CC(C=O)C2

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.53
CHRM1 P11229 4/20 0.53
CHRM3 P20309 4/20 0.53
DRD2 P14416 4/20 0.51
DRD3 P35462 4/20 0.51
DRD4 P21917 3/20 0.51
HTR1A P08908 2/20 0.49
CYP19A1 P11511 1/20 0.47
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27394377 0.82 ADRA1A (0.55) CHRM2CHRM1CHRM3DRD2
SCHEMBL27469141 0.77 ACHE (0.40) CHRM2CHRM1CHRM3DRD2DRD3
SCHEMBL7606129 0.77 DRD2 (0.57) CHRM2CHRM1CHRM3DRD2DRD3
SCHEMBL17682886 0.75 HTR1A (0.51) CHRM2CHRM1CHRM3DRD2DRD3
SCHEMBL27390763 0.74 ALDH1A1 (0.49)
SCHEMBL24029258 0.74 DRD2 (0.54) CHRM2CHRM1CHRM3DRD2DRD3
SCHEMBL31324598 0.74 DRD2 (0.73) CHRM2CHRM1CHRM3DRD2DRD3
SCHEMBL14545524 0.74 DRD2 (0.54) CHRM2CHRM1CHRM3DRD2DRD3
SCHEMBL16482975 0.74 DRD2 (0.54) CHRM2CHRM1CHRM3DRD2DRD3
SCHEMBL23856659 0.74 HTR1A (0.38) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422134-B1 5-HT SELECTIVE AGENTS ABBOTT LAB (US) 1996-06-12 EP disclosed
US-5244888-A Hexahydroindenopyrroles and hexahydrobenzisoindoles ABBOTT LABORATORIES (US) 1993-09-14 US disclosed
US-5049564-A Hypotensive, 5-hydroxytryptamine ABBOTT LABORATORIES (US) 1991-09-17 US disclosed
EP-0422134-A1 5-HT SELECTIVE AGENTS. ABBOTT LAB (US) 1991-04-17 EP disclosed
WO-1990006927-A1 5-HT SELECTIVE AGENTS ABBOTT LABORATORIES (US) 1990-06-28 WO disclosed