SCHEMBL9037405

SCHEMBL9037405

CC(C)Nc1cccnc1N1CCN(C(=O)c2c[nH]c3cc(CN(C)C)ccc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
CHRM1 P11229 1/20 0.48
MAOA P21397 1/20 0.48
TBXA2R P21731 1/20 0.48
OPRM1 P35372 1/20 0.48
MDH1 P40925 1/20 0.48
KCNH2 Q12809 1/20 0.48
ABCG2 Q9UNQ0 1/20 0.48
AVPR1A P37288 4/20 0.41
SSTR2 P30874 7/20 0.39
GFER P55789 1/20 0.39
HDAC1 Q13547 3/20 0.38
HDAC6 Q9UBN7 3/20 0.38
CHRM2 P08172 1/20 0.38
HTT P42858 1/20 0.37
MAPK14 Q16539 1/20 0.37
IDH1 O75874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038924 0.91 ADRA2A (0.49) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL9036880 0.87 ADRA2A (0.49) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL9037304 0.85 ADRA2A (0.51) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL9037017 0.85 ADRA2A (0.50) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL9037801 0.84 GFER (0.55) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL9038780 0.84 ADRA2A (0.49) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL9038099 0.84 ADRA2A (0.49) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL9035802 0.83 ADRA2A (0.49) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL8795126 0.83 ADRA2A (0.48) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL9037435 0.81 ADRA2A (0.50) ADRA2AADORA3CHRM1MAOATBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP claimed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO claimed