SCHEMBL9038872

SCHEMBL9038872

CC(C)n1cccc1C(=O)NCCC(=O)O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
MME P08473 1/20 0.40
ACE P12821 1/20 0.40
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GCG P01275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9039943 0.82 CYP3A4 (0.40) NPC1RAB9AL3MBTL1CYP1A2CYP3A4
SCHEMBL6988127 0.80 RAB9A (0.68) NPC1RAB9AL3MBTL1CYP2C9
SCHEMBL6993812 0.78 NPC1 (0.47) NPC1RAB9AMMEACELMNA
SCHEMBL9037906 0.75 NPC1 (0.48) NPC1RAB9ALMNAL3MBTL1NPSR1
SCHEMBL1664507 0.73 CYP1A2 (0.44) NPC1RAB9AL3MBTL1CYP1A2CYP3A4
SCHEMBL9037774 0.73 NPSR1 (0.47) NPC1RAB9ALMNANPSR1ITGB3
SCHEMBL6992210 0.72 CNR2 (0.64) NPC1RAB9AMMEACE
SCHEMBL26205734 0.69 MAPK1 (0.43) NPC1RAB9ALMNACA1CA2
SCHEMBL6796081 0.69 LMNA (0.40) LMNAL3MBTL1CYP1A2CYP3A4CYP2C9
SCHEMBL1520499 0.67 L3MBTL1 (0.61) NPC1RAB9ALMNAL3MBTL1ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441349-B1 Pyrroloazepine derivatives SUNTORY LTD (JP) 1996-01-03 EP disclosed
US-5416082-A Antiserotonine agents SUNTORY LIMITED (JP) 1995-05-16 US disclosed
US-5391731-A Useful therapeutics for circulatory diseases SUNTORY LIMITED (JP) 1995-02-21 US disclosed
US-5206239-A Cardiovascular disorders SUNTORY LIMITED (JP) 1993-04-27 US disclosed
EP-0441349-A1 Pyrroloazepine derivatives SUNTORY LIMITED (JP) 1991-08-14 EP disclosed