SCHEMBL9039665

SCHEMBL9039665

COc1ccc2c(c1)c(CCCN1CCCC1CC(=O)c1ccc(F)cc1)cn2C

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.46
MTNR1B P49286 5/20 0.46
NQO2 P16083 1/20 0.46
ADRB2 P07550 4/20 0.44
AKR1C3 P42330 2/20 0.43
HTR6 P50406 2/20 0.42
HRH3 Q9Y5N1 3/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
AKR1C2 P52895 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310519 0.83 NQO2 (0.46) MTNR1AMTNR1BNQO2ADRB2AKR1C3
Hydrochloric Acid SCHEMBL8912255 0.82 NQO2 (0.45) MTNR1AMTNR1BNQO2ADRB2AKR1C3
SCHEMBL8307225 0.79 NQO2 (0.47) MTNR1AMTNR1BNQO2ADRB2AKR1C3
Hydrochloric Acid SCHEMBL8913070 0.79 NQO2 (0.46) MTNR1AMTNR1BNQO2ADRB2AKR1C3
SCHEMBL31670925 0.69 HTR1B (0.63) MTNR1AMTNR1BNQO2ADRB2HTR6
SCHEMBL8304470 0.68 ADRB2 (0.70) MTNR1AMTNR1BNQO2ADRB2HTR6
SCHEMBL11343620 0.68 KDM2B (0.52) ALDH1A1KDM4ECYP3A4CYP2D6
SCHEMBL11521240 0.67 AKR1C3 (0.56) AKR1C3LMNAAKR1C2CYP2D6
SCHEMBL8306860 0.67 HTR1A (0.62)
SCHEMBL18509701 0.66 MTNR1A (0.67) MTNR1AMTNR1BNQO2ADRB2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747379-A1 Derivatives of indole, indazole and benzisoxazole for the treatment of schizophrenia ADIR ET COMPAGNIE (FR) 1996-12-11 EP disclosed