SCHEMBL8307225

SCHEMBL8307225

COc1ccc2c(c1)c(CCN1CCC(CC(=O)c3ccc(F)cc3)C1)cn2C

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.47
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
ADRB2 P07550 1/20 0.45
HTR1A P08908 1/20 0.45
SLC6A4 P31645 1/20 0.45
DRD2 P14416 2/20 0.44
HTR2A P28223 2/20 0.44
HTR2C P28335 2/20 0.44
HTR2B P41595 2/20 0.44
SIGMAR1 Q99720 2/20 0.44
AKR1C3 P42330 1/20 0.44
HTR6 P50406 2/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8913070 0.99 NQO2 (0.46) NQO2MTNR1AMTNR1BADRB2HTR1A
SCHEMBL8310519 0.95 NQO2 (0.46) NQO2MTNR1AMTNR1BADRB2HTR1A
Hydrochloric Acid SCHEMBL8912255 0.94 NQO2 (0.45) NQO2MTNR1AMTNR1BADRB2HTR1A
SCHEMBL8306212 0.83 HTR2A (0.55) HTR1ASLC6A4DRD2HTR2A
Hydrochloric Acid SCHEMBL9073679 0.83 HTR2A (0.54) HTR1ASLC6A4DRD2HTR2A
SCHEMBL9039665 0.79 MTNR1A (0.46) NQO2MTNR1AMTNR1BADRB2AKR1C3
SCHEMBL8306860 0.79 HTR1A (0.62) HTR1ASLC6A4DRD2
SCHEMBL32669268 0.72 ADRB2 (0.67) NQO2MTNR1AMTNR1BADRB2HTR2A
SCHEMBL9870723 0.72 DRD2 (0.65) HTR1ADRD2HTR2AHTR2CHTR2B
SCHEMBL8916558 0.70 DRD2 (0.40) DRD2HTR2AHTR2CHTR2BSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747379-B1 Derivatives of indole, indazole and benzisoxazole for the treatment of schizophrenia ADIR (FR) 1999-08-11 EP disclosed
US-5703070-A PSYCHOLOGICAL DISORDERS ADIR ET COMPAGNIE (FR) 1997-12-30 US disclosed
EP-0747379-A1 Derivatives of indole, indazole and benzisoxazole for the treatment of schizophrenia ADIR ET COMPAGNIE (FR) 1996-12-11 EP disclosed