SCHEMBL9040202

SCHEMBL9040202

CCCCOc1ccc(-c2nc3ccccc3n2Cc2ccc(-c3ccccc3OC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.57
DRD3 P35462 5/20 0.57
PDE6D O43924 4/20 0.52
AGTR2 P50052 2/20 0.51
HTT P42858 3/20 0.51
KDM4E B2RXH2 2/20 0.51
LMNA P02545 2/20 0.51
ALDH1A1 P00352 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
CNR2 P34972 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
PIN1 Q13526 2/20 0.49
ESR1 P03372 1/20 0.49
TP53 P04637 2/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
AGTR1 P30556 1/20 0.47
TBXA2R P21731 1/20 0.47
PPARG P37231 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9041371 0.90 PDE6D (0.54) DRD2DRD3PDE6DHTTKDM4E
SCHEMBL9040832 0.90 DRD2 (0.60) DRD2DRD3PDE6DAGTR2HTT
SCHEMBL9042322 0.90 KDM4E (0.66) DRD2PDE6DHTTKDM4ELMNA
SCHEMBL9043441 0.89 TP53 (0.56) DRD2PDE6DAGTR2HTTKDM4E
SCHEMBL9041081 0.88 ALDH1A1 (0.51) DRD2DRD3PDE6DAGTR2HTT
SCHEMBL8397011 0.87 DRD2 (0.58) DRD2DRD3PDE6DAGTR2HTT
SCHEMBL9041236 0.84 AGTR1 (0.66) AGTR2AGTR1PPARG
SCHEMBL9040419 0.84 HDAC1 (0.52) DRD2AGTR2HTTAGTR1TBXA2R
SCHEMBL9043424 0.83 GRM2 (0.53) DRD2PDE6DHTTKDM4ELMNA
SCHEMBL9043483 0.83 PPARG (0.67) AGTR2AGTR1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0392317-B1 Benzimidazoles, drugs containing these compounds and process for their preparation THOMAE GMBH DR K (DE) 1996-01-03 EP disclosed
EP-0392317-A2 Benzimidazoles, drugs containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1990-10-17 EP disclosed