SCHEMBL9040489

SCHEMBL9040489

Cc1ccccc1NC(=O)NC1C=C(c2ccccc2)c2ccccc2N(CC(=O)OC(C)(C)C)C1=O

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 10/20 0.47
HDAC3 O15379 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
CCKAR P32238 1/20 0.40
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
BRD4 O60885 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9041968 0.90 CCKBR (0.50) CCKBRHDAC3HDAC1HDAC8HDAC6
SCHEMBL9039747 0.90 CCKBR (0.51) CCKBRHDAC3HDAC1HDAC8HDAC6
SCHEMBL9040362 0.89 CCKBR (0.52) CCKBRCCKARCYP3A4MAPTTSHR
SCHEMBL9040311 0.88 CCKBR (0.51) CCKBRCCKAR
SCHEMBL9039449 0.88 ALDH1A1 (0.46) CCKBRCCKARCYP3A4MAPTTSHR
SCHEMBL9039719 0.87 CCKBR (0.58) CCKBRCCKARCYP3A4MAPTTSHR
SCHEMBL9038073 0.85 CYP3A4 (0.53) CCKBRCCKARCYP3A4MAPTTSHR
SCHEMBL9040062 0.85 CCKBR (0.62) CCKBRCCKARCYP3A4MAPTTSHR
SCHEMBL9039585 0.85 CCKBR (0.61) CCKBR
SCHEMBL9041035 0.84 CCKBR (0.51) CCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0703222-A1 3-AMINOAZEPINE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-03-27 EP disclosed