SCHEMBL9040678

SCHEMBL9040678

Clc1cc(-c2nnn[nH]2)n(-c2ccc(Cn3cnc4cccnc43)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
TP53 P04637 1/20 0.46
PABPC1 P11940 1/20 0.46
CSF1R P07333 6/20 0.39
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 1/20 0.35
GRM2 Q14416 1/20 0.35
POLB P06746 2/20 0.34
GABRP O00591 2/20 0.33
GABRD O14764 2/20 0.33
GABRA1 P14867 2/20 0.33
GABRB1 P18505 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA5 P31644 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9042834 0.80 AGTR1 (0.50) MEN1KMT2ATP53MAPT
SCHEMBL9040754 0.79 AGTR1 (0.51) MEN1KMT2ATP53MAPT
SCHEMBL7472677 0.74 RAB9A (0.36) HTTSMN1; SMN2MAPT
SCHEMBL13508712 0.74 TP53 (0.68) MEN1KMT2ATP53PABPC1CSF1R
SCHEMBL9040197 0.72 AGTR1 (0.42) HTR1A
SCHEMBL7469162 0.72 POLB (0.36) MEN1KMT2ATP53HTTSMN1; SMN2
SCHEMBL7464057 0.71 AGTR1 (0.50)
SCHEMBL9310709 0.71 AGTR2 (0.38)
SCHEMBL9041166 0.71 AGTR2 (0.51)
SCHEMBL7467991 0.71 NR1H4 (0.38) TP53HTTSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0480204-B1 Imidazole derivatives, potent and selective antagonists of angiotensin II receptor FUJISAWA PHARMACEUTICAL CO (JP) 1996-03-20 EP disclosed
US-5215994-A Treating or preventing hypertension or heart failure FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-06-01 US disclosed
US-5210092-A Hypotensive agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-11 US disclosed
EP-0480204-A1 Imidazole derivatives, potent and selective antagonists of angiotensin II receptor FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-15 EP disclosed