SCHEMBL9040830

SCHEMBL9040830

CN1CCC(=O)c2ccn(CCCCN3CCC(Cc4ccccc4)CC3)c2C1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.52
SIGMAR1 Q99720 3/20 0.51
CCR3 P51677 3/20 0.51
ADRB2 P07550 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
ADRB1 P08588 1/20 0.46
CHRM5 P08912 1/20 0.46
CHRM1 P11229 1/20 0.46
DRD2 P14416 1/20 0.46
CHRM3 P20309 1/20 0.46
DRD4 P21917 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
DRD3 P35462 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
TMEM97 Q5BJF2 1/20 0.46
HRH3 Q9Y5N1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9039006 0.85 SIGMAR1 (0.47) SIGMAR1CHRM2CHRM4CHRM5CHRM1
SCHEMBL6988906 0.85 HTR1A (0.47) CCR3
SCHEMBL9042911 0.82 KCNH2 (0.55) KCNH2DRD2HRH3
SCHEMBL9040406 0.81 BCHE (0.50) KCNH2CHRM2CHRM4ADRB1CHRM5
SCHEMBL6986161 0.81 HTR1A (0.53) KCNH2SIGMAR1DRD2DRD4DRD3
SCHEMBL9266055 0.80 HTR1A (0.54) KCNH2DRD2DRD4DRD3
SCHEMBL6988888 0.79 DRD2 (0.57) DRD2ADRA1BDRD3
SCHEMBL9038772 0.79 KCNH2 (0.48) KCNH2DRD2ADRA1DADRA1AADRA1B
SCHEMBL9580851 0.78 KCNH2 (0.47) KCNH2ADRB2CHRM2CHRM4ADRB1
SCHEMBL6991322 0.78 SIGMAR1 (0.51) KCNH2SIGMAR1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441349-B1 Pyrroloazepine derivatives SUNTORY LTD (JP) 1996-01-03 EP disclosed
US-5416082-A Antiserotonine agents SUNTORY LIMITED (JP) 1995-05-16 US disclosed
US-5391731-A Useful therapeutics for circulatory diseases SUNTORY LIMITED (JP) 1995-02-21 US disclosed
US-5206239-A Cardiovascular disorders SUNTORY LIMITED (JP) 1993-04-27 US disclosed
EP-0441349-A1 Pyrroloazepine derivatives SUNTORY LIMITED (JP) 1991-08-14 EP disclosed