SCHEMBL9040983

SCHEMBL9040983

Cc1sc2ncc([N+](=O)[O-])c(-c3ccccc3Cl)c2c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.36
PIN1 Q13526 3/20 0.35
HSD11B1 P28845 1/20 0.35
ALDH1A1 P00352 5/20 0.35
KDM4E B2RXH2 4/20 0.35
TDP1 Q9NUW8 2/20 0.35
LMNA P02545 4/20 0.34
HTT P42858 3/20 0.34
MAPK1 P28482 2/20 0.34
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 3/20 0.34
HPGD P15428 3/20 0.34
MRGPRX1 Q96LB2 2/20 0.34
POLB P06746 1/20 0.34
NLRP3 Q96P20 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9041404 0.79 LIMK1 (0.41) ALDH1A1KDM4ETDP1LMNAHTT
SCHEMBL9040652 0.79 HSD11B1 (0.37) PKMPIN1HSD11B1ALDH1A1KDM4E
SCHEMBL9042985 0.77 MAPT (0.46) ALDH1A1KDM4ELMNAHTTMAPK1
SCHEMBL9041501 0.77 ALDH1A1 (0.43) ALDH1A1KDM4ETDP1LMNAHTT
SCHEMBL9158252 0.76 MAPT (0.40) PKMPIN1HSD11B1ALDH1A1KDM4E
SCHEMBL9042591 0.74 SELE (0.40) ALDH1A1KDM4ELMNAHTTRAB9A
SCHEMBL9164973 0.73 POLB (0.44) PKMPIN1ALDH1A1KDM4ETDP1
SCHEMBL9163731 0.72 HSD11B1 (0.38) PKMPIN1HSD11B1ALDH1A1KDM4E
SCHEMBL9163609 0.72 HSD11B1 (0.39) PKMPIN1HSD11B1ALDH1A1KDM4E
SCHEMBL9159576 0.71 MAPT (0.40) PKMPIN1HSD11B1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0472116-B1 Thienopyridine Derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-01-31 EP disclosed
US-5256782-A For anticholesterol agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-10-26 US disclosed
US-5143919-A Acyl-CoA:cholesterol acyltransferase inhibitors; anticholesterol agents; TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-09-01 US disclosed
EP-0472116-A1 Thienopyridine Derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1992-02-26 EP disclosed