SCHEMBL904138

SCHEMBL904138

C[S+]([O-])c1ccc(Br)cc1F

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.37
KDM1A O60341 2/20 0.35
KDM1B Q8NB78 1/20 0.35
PYCR1 P32322 1/20 0.33
NPC1 O15118 4/20 0.33
RAB9A P51151 4/20 0.33
NMT1 P30419 1/20 0.33
AKR1B1 P15121 1/20 0.32
APLNR P35414 2/20 0.31
ALDH1A1 P00352 2/20 0.30
ALOX12 P18054 2/20 0.30
LMNA P02545 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
TP53 P04637 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31426534 0.85 DGAT1 (0.34) DGAT1KDM1AKDM1BPYCR1NPC1
SCHEMBL777155 0.78 ALDH1A1 (0.39) ALDH1A1ALOX12
SCHEMBL19409342 0.78 ALOX15 (0.39) PYCR1ALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL13461896 0.77 NFE2L2 (0.35) AKR1B1SMN1; SMN2TP53
SCHEMBL20149232 0.75 ALDH1A1 (0.33) ALDH1A1LMNA
SCHEMBL11855535 0.75
SCHEMBL18921866 0.75 CYP2A6 (0.33) ALDH1A1
SCHEMBL31090434 0.75 CYP2A6 (0.33) ALDH1A1
SCHEMBL28779497 0.73 CYP2A6 (0.38)
SCHEMBL27348288 0.72 ALDH1A1 (0.33) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed