SCHEMBL9041817

SCHEMBL9041817

Nc1nc(N)c2c(n1)NCC2CCNc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MTHFD1 P11586 1/20 0.59
SOST Q9BQB4 1/20 0.55
ATIC P31939 3/20 0.53
DHFR P00374 2/20 0.52
GART P22102 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9220611 0.97 MTHFD1 (0.56) MTHFD1SOSTATICDHFRGART
SCHEMBL9220625 0.90 MTHFD1 (0.49) MTHFD1SOSTATICDHFRGART
SCHEMBL8997257 0.86 GART (0.61) ATICDHFRGART
SCHEMBL8997170 0.85 DHFR (0.55) ATICDHFRGART
SCHEMBL9042931 0.85 DHFR (0.60) ATICDHFRGART
SCHEMBL9758306 0.85 DHFR (0.55) ATICDHFRGART
SCHEMBL9043308 0.85 DHFR (0.57) ATICDHFRGART
SCHEMBL9088274 0.85 ATIC (0.51) MTHFD1ATICDHFRGART
SCHEMBL9041616 0.85 GART (0.54) MTHFD1ATICGART
SCHEMBL8571393 0.84 ATIC (0.59) MTHFD1ATICDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0400562-B1 Pyrrolopyrimidines, their production and use as tumoricidal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-08-21 EP disclosed