SCHEMBL9043231

SCHEMBL9043231

O=C(O)Oc1cn2c(n1)c(=O)[nH]c1ccccc12

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.48
ADORA3 P0DMS8 9/20 0.44
PARP1 P09874 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
G6PD P11413 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
ALOX12 P18054 1/20 0.42
HKDC1 Q2TB90 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ADORA1 P30542 3/20 0.41
ADORA2A P29274 2/20 0.41
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7507051 0.80 POLB (0.51) POLBADORA3PARP1KDM4EALDH1A1
SCHEMBL7773136 0.80 GRIA1 (0.51)
SCHEMBL9256388 0.75 ADORA3 (0.55) POLBADORA3PARP1KDM4EALDH1A1
SCHEMBL7269351 0.75 POLB (0.55) POLBADORA3PARP1KDM4EALDH1A1
SCHEMBL8557963 0.73 GRIN2D (0.40)
SCHEMBL30748698 0.73 ADORA3 (0.61) POLBADORA3MEN1KMT2A
SCHEMBL7517896 0.73 ADORA3 (0.61) POLBADORA3MEN1KMT2A
SCHEMBL8553821 0.72 POLB (0.49) POLBADORA3KDM4EALDH1A1MAPT
SCHEMBL28887969 0.70 ADORA1 (0.49) POLBADORA3ADORA1ADORA2A
SCHEMBL8555309 0.69 ADORA3 (0.47) POLBADORA3KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691970-A1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 1996-01-17 EP disclosed
WO-1994022865-A1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 1994-10-13 WO disclosed