SCHEMBL9044339

SCHEMBL9044339

O=C(O)C1CN(Cc2ccncc2)C(=O)C1=O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
GRM2 Q14416 1/20 0.40
KDM4E B2RXH2 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HDAC1 Q13547 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ARG1 P05089 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
CACNA1I Q9P0X4 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
NPC1 O15118 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
BLM P54132 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9043612 0.86 POLB (0.46) ALDH1A1KMT2AHTTSMN1; SMN2CYP2C9
SCHEMBL9044246 0.82 HTT (0.42) ALDH1A1KDM4EMEN1KMT2AHDAC1
SCHEMBL9043025 0.81 ALDH1A1 (0.55) ALDH1A1GRM2KDM4EMEN1KMT2A
SCHEMBL9042078 0.79 GRM5 (0.47) ALDH1A1MEN1KMT2ASMN1; SMN2SIGMAR1
SCHEMBL9042862 0.76 L3MBTL1 (0.50) ALDH1A1KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL7462557 0.73 ALDH1A1 (0.71) ALDH1A1HTTSMN1; SMN2
SCHEMBL9043663 0.71 L3MBTL1 (0.46) ALDH1A1HTTSMN1; SMN2
SCHEMBL11492920 0.71 FKBP1A (0.48) ALDH1A1MEN1KMT2ASMN1; SMN2CYP2C9
SCHEMBL9045382 0.71 KDM4E (0.39) ALDH1A1GRM2KDM4EMEN1KMT2A
SCHEMBL14829141 0.71 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0553130-B1 PYRROLIDINE DIONE DERIVATIVES PFIZER (US) 1996-01-03 EP claimed