SCHEMBL9044800

SCHEMBL9044800

COc1ccc(OCCOc2ccc(C(=O)C(=O)O)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.62
CES1 P23141 2/20 0.62
MAPT P10636 6/20 0.62
PTPRC P08575 4/20 0.59
PTPN1 P18031 4/20 0.59
PTPN2 P17706 1/20 0.59
PTPRF P10586 1/20 0.57
RAB9A P51151 2/20 0.56
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
NPC1 O15118 1/20 0.54
POLB P06746 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
LMNA P02545 3/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
PKM P14618 1/20 0.53
MTNR1A P48039 1/20 0.51
MTNR1B P49286 1/20 0.51
TP53 P04637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9043540 0.91 PTPRC (0.69) MAPTPTPRCPTPN1PTPN2PTPRF
SCHEMBL9042648 0.89 PTPRC (0.59) CES2CES1MAPTPTPRCPTPN1
SCHEMBL9043116 0.89 KDM4E (0.57) CES2CES1MAPTPTPRCPTPN1
SCHEMBL906482 0.89 CES2 (0.78) CES2CES1MAPTPTPRCPTPN1
SCHEMBL9044645 0.86 L3MBTL1 (0.61) CES2CES1MAPTPTPRCPTPN1
SCHEMBL9044396 0.85 PKM (0.72) MAPTPTPRCPTPN1PTPN2PTPRF
SCHEMBL9043716 0.84 MAPT (0.56) MAPTPTPRCPTPN1PTPN2PTPRF
SCHEMBL9042386 0.84 MAPT (0.61) CES2CES1MAPTRAB9ACA1
SCHEMBL16917421 0.84 TP53 (0.67) PTPRCPTPN1PTPN2PTPRFL3MBTL1
SCHEMBL9042263 0.83 MAPT (0.56) MAPTPTPRCPTPN1PTPN2PTPRF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512352-B1 Substituted carboxylic acid derivatives HOFFMANN LA ROCHE (CH) 1996-03-27 EP disclosed
US-5344843-A Carnitine acryltransferase enzyme inhibitors as antiischemic agents and for cardiovascular disorders HOFFMAN-LA ROCHE INC. (US) 1994-09-06 US disclosed
EP-0512352-A2 Substituted carboxylic acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-11-11 EP disclosed