SCHEMBL9045256

SCHEMBL9045256

COC(=O)c1ccc(CCn2c(C)nc3nc(C(=O)C(C)(C)C)cc-3c2O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
MAPT P10636 3/20 0.38
TP53 P04637 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
CKS1B P61024 1/20 0.38
SKP2 Q13309 1/20 0.38
HIF1A Q16665 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP4A11 Q02928 2/20 0.38
TLR7 Q9NYK1 1/20 0.38
DRD2 P14416 3/20 0.37
TBXA2R P21731 3/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045295 0.68 GAA (0.43) KDM4EMAPTTP53CYP1A2CYP3A4
SCHEMBL9045449 0.67 YTHDC1 (0.39) KDM4ETP53CYP1A2CYP3A4CYP2C9
SCHEMBL1426221 0.66 ALDH1A1 (0.49) KDM4EMAPTTP53CYP1A2CYP3A4
SCHEMBL1426809 0.65 CYP4A11 (0.49) KDM4EMAPTTP53CYP1A2CYP3A4
SCHEMBL1426725 0.65 CYP4A11 (0.49) KDM4EMAPTTP53CYP1A2CYP3A4
SCHEMBL12734653 0.65 CYP1A2 (0.48) KDM4EMAPTTP53CYP1A2CYP3A4
SCHEMBL3526493 0.63 LMNA (0.56) KDM4EMAPTTP53DRD2TBXA2R
SCHEMBL70185 0.63 CYP4A11 (0.75) KDM4EMAPTTP53CYP1A2CYP3A4
SCHEMBL1426040 0.63 CYP1A2 (0.47) KDM4EMAPTTP53CYP1A2CYP3A4
SCHEMBL1003052 0.63 HDAC6 (0.68) CYP4A11DRD2TBXA2RRAB9ACYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed