SCHEMBL9045658

SCHEMBL9045658

COC(=O)CC[C@H](NC(=O)c1ccc(CCn2cnc3nc(NC(=O)C(C)(C)C)cc-3c2O)cc1F)C(=O)OC

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ATIC P31939 3/20 0.36
SHMT1 P34896 3/20 0.36
SHMT2 P34897 3/20 0.36
GART P22102 3/20 0.35
MAPK14 Q16539 1/20 0.32
FOLR2 P14207 2/20 0.32
FOLR1 P15328 2/20 0.32
SLC46A1 Q96NT5 2/20 0.32
SLC19A1 P41440 1/20 0.32
MAPK1 P28482 2/20 0.32
ALDH1A1 P00352 1/20 0.32
KDR P35968 2/20 0.32
CNR2 P34972 3/20 0.31
TYMS P04818 2/20 0.31
CNR1 P21554 1/20 0.31
CSNK1D P48730 1/20 0.30
CSNK1E P49674 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045922 0.90 TAS1R3 (0.35) MAPK14ALDH1A1
SCHEMBL9044079 0.87 MAPK14 (0.36) MAPK14FOLR2FOLR1SLC46A1ALDH1A1
SCHEMBL9777813 0.86 ALDH1A1 (0.34) MAPK1ALDH1A1
SCHEMBL9045652 0.85 MAPK14 (0.32) MAPK14MAPK1ALDH1A1KDR
SCHEMBL9046657 0.83 ATIC (0.34) ATICSHMT1SHMT2GARTMAPK14
SCHEMBL9044092 0.83 MAPK14 (0.32) MAPK14MAPK1ALDH1A1KDR
SCHEMBL9047978 0.82 KMT2A (0.36)
SCHEMBL9044865 0.81 KMT2A (0.37)
SCHEMBL9047324 0.81 KMT2A (0.37)
SCHEMBL9045286 0.79 ADORA1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
US-5344932-A N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives TRUSTEES OF PRINCETON UNIVERSITY (US) 1994-09-06 US disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed