SCHEMBL9045922

SCHEMBL9045922

COC(=O)CC[C@H](NC(=O)c1ccc(CCn2cnc3nc(NC(=O)C(C)(C)C)cc-3c2O)cc1)C(=O)OC

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
ROCK2 O75116 1/20 0.35
MAPK14 Q16539 2/20 0.34
LNPEP Q9UIQ6 4/20 0.33
ERAP2 Q6P179 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
ERAP1 Q9NZ08 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045658 0.90 ATIC (0.36) MAPK14ALDH1A1
SCHEMBL9777813 0.90 ALDH1A1 (0.34) TAS1R3TAS1R1ALDH1A1CA12CA1
SCHEMBL9044079 0.89 MAPK14 (0.36) TAS1R3TAS1R1L3MBTL1ROCK2MAPK14
SCHEMBL9043718 0.87 ATIC (0.43)
SCHEMBL9046657 0.87 ATIC (0.34) MAPK14ALDH1A1HPGDCA12CA1
SCHEMBL9471199 0.86 TAS1R3 (0.41) TAS1R3TAS1R1L3MBTL1ROCK2MAPK14
SCHEMBL9047978 0.86 KMT2A (0.36) CA12CA1CA2CA9
SCHEMBL9044865 0.85 KMT2A (0.37) CA12CA1CA2CA9
SCHEMBL9047324 0.85 KMT2A (0.37) CA12CA1CA2CA9
SCHEMBL9046201 0.83 TAS1R3 (0.41) TAS1R3TAS1R1L3MBTL1ROCK2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
US-5344932-A N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives TRUSTEES OF PRINCETON UNIVERSITY (US) 1994-09-06 US disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed