SCHEMBL9045676

SCHEMBL9045676

C1=CCC2=c3nc(CC4CCCN(Cc5ccccc5)C4)sc3=CC2=C1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.40
CCR1 P32246 1/20 0.39
CCR3 P51677 1/20 0.39
CYP2D6 P10635 3/20 0.39
CARM1 Q86X55 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
CYP3A4 P08684 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ACHE P22303 2/20 0.37
ACKR3 P25106 1/20 0.37
MAOB P27338 1/20 0.36
CYP2C9 P11712 2/20 0.36
PDE8B O95263 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9049957 0.98 BCHE (0.39) BCHECCR1CCR3CYP2D6CARM1
SCHEMBL9046919 0.94 DRD2 (0.40) BCHECCR3CYP2D6CARM1PRMT6
Hydrochloric Acid SCHEMBL9050368 0.93 DRD2 (0.39) BCHECCR3CYP2D6CARM1PRMT6
SCHEMBL9047841 0.80 ACHE (0.37) BCHECYP2D6CYP3A4CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL9045686 0.79 ACHE (0.37) BCHECYP2D6CYP3A4CYP1A2CYP2C19
SCHEMBL9047832 0.73 HRH3 (0.33)
SCHEMBL9047746 0.71 L3MBTL1 (0.37) CYP2D6CYP3A4CYP1A2ALDH1A1
SCHEMBL9047634 0.70 DRD3 (0.35) DRD2DRD4DRD3
SCHEMBL9045662 0.69 BCHE (0.44) BCHECCR1CCR3CYP2D6CARM1
SCHEMBL8238364 0.69 BCHE (0.70) BCHECCR3CYP2D6CARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749966-A1 5-HT 3 RECEPTOR AGONIST, NOVEL THIAZOLE DERIVATIVE, AND INTERMEDIATE THEREFOR YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-12-27 EP disclosed