SCHEMBL9046000

SCHEMBL9046000

O=C(O)c1cc(=O)c2ccc(F)cc2n1-c1ccccc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NOTUM Q6P988 1/20 0.43
MPI P34949 1/20 0.41
MAT2A P31153 1/20 0.40
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
ATM Q13315 1/20 0.38
MAPK8 P45983 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GLA P06280 1/20 0.38
TSHR P16473 1/20 0.37
HSP90AA1 P07900 1/20 0.37
LMNA P02545 1/20 0.37
MAOB P27338 1/20 0.37
POLB P06746 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9044837 0.92 GLA (0.40) KDM4ESMN1; SMN2NOTUMMAT2AALDH1A1
SCHEMBL9046545 0.86 NOTUM (0.44) KDM4ESMN1; SMN2NOTUMALDH1A1HSD17B10
SCHEMBL9044266 0.83 TDP1 (0.44) KDM4ENOTUMMPIMAT2AALDH1A1
SCHEMBL9046534 0.81 NOTUM (0.41) KDM4ESMN1; SMN2NOTUMMAT2AALDH1A1
SCHEMBL10445661 0.78 GLA (0.37) KDM4EMAT2AALDH1A1HPGDHSD17B10
Bicarbonate SCHEMBL9046002 0.77 MAPK8 (0.47) KDM4ESMN1; SMN2MPIATMMAPK8
SCHEMBL12984605 0.70 ALDH1A1 (0.63) KDM4EALDH1A1HPGDHSD17B10ATM
SCHEMBL26596771 0.66 ATM (0.58) KDM4EMPIMAT2AALDH1A1ATM
SCHEMBL14575936 0.66 CAPN1 (0.53) ATMMAPK8
SCHEMBL5824022 0.66 HPGD (0.41) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422485-B1 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1996-04-03 EP disclosed
US-5300643-A Viricides BAYER AKTIENGESELLSCHAFT (DE) 1994-04-05 US disclosed
US-5217972-A QUINOLONECARBOXYLIC ACID DERIVATIVES AND THEIR USE AS ANTIVIRAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1993-06-08 US disclosed
EP-0422485-A2 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1991-04-17 EP disclosed