Bicarbonate

Bicarbonate

SCHEMBL9046002

O=C(O)O.O=c1ccn(-c2ccccc2F)c2cc(F)ccc12

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 7/20 0.47
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
ATM Q13315 1/20 0.40
MPI P34949 1/20 0.40
RORC P51449 2/20 0.39
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
SCN2B O60939 1/20 0.37
SCN1B Q07699 1/20 0.37
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
KDM4E B2RXH2 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CD74 P04233 1/20 0.36
MIF P14174 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL9044839 0.89 HTR1A (0.38) MAPK8ATMRORCCYP3A4CYP2C9
Bicarbonate SCHEMBL9046548 0.86 PTGS1 (0.43) MAPK8PTGS1PTGS2RORCMAPT
Bicarbonate SCHEMBL9046542 0.83 PTGS1 (0.41) MAPK8PTGS1PTGS2RORCSCN2B
Bicarbonate SCHEMBL9044272 0.80 RORC (0.47) RORCMAPTKDM4ESMN1; SMN2CYP3A4
SCHEMBL339069 0.79 KDM4E (0.44) PTGS1PTGS2RORCSCN2BSCN1B
SCHEMBL14575936 0.78 CAPN1 (0.53) MAPK8ATM
SCHEMBL9046000 0.77 KDM4E (0.43) MAPK8ATMMPITP53MAPT
SCHEMBL14576338 0.74 ATM (0.51) MAPK8ATMMPIMAPTSCN2B
SCHEMBL10593432 0.73 GLA (0.35) PTGS2ATM
SCHEMBL16464113 0.72 NR1I2 (0.43) ATMTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422485-B1 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1996-04-03 EP disclosed
EP-0422485-A2 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1991-04-17 EP disclosed