SCHEMBL9044837

SCHEMBL9044837

O=C(O)c1cc(=O)c2ccc(F)cc2n1-c1ccc(F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.40
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PTGS1 P23219 2/20 0.35
PTGS2 P35354 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
MAT2A P31153 1/20 0.34
NOTUM Q6P988 1/20 0.34
GRM5 P41594 1/20 0.34
MEN1 O00255 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
CCR2 P41597 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9046000 0.92 KDM4E (0.43) GLAALDH1A1KDM4EHPGDHSD17B10
SCHEMBL10445661 0.86 GLA (0.37) GLAALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9044266 0.83 TDP1 (0.44) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL9046545 0.77 NOTUM (0.44) ALDH1A1KDM4EHSD17B10PTGS1PTGS2
Bicarbonate SCHEMBL9044839 0.73 HTR1A (0.38) GLAL3MBTL1MEN1KMT2AEPHA2
SCHEMBL9046534 0.73 NOTUM (0.41) ALDH1A1KDM4EHSD17B10SMN1; SMN2MAPT
SCHEMBL14354361 0.70 ALDH1A1 (0.42) GLAALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL14354357 0.70 GLA (0.41) GLAPTGS1PTGS2L3MBTL1
Bicarbonate SCHEMBL9046002 0.69 MAPK8 (0.47) KDM4EPTGS1PTGS2SMN1; SMN2MAPT
SCHEMBL9147090 0.69 EPHA2 (0.53) ALDH1A1KDM4EHPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422485-B1 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1996-04-03 EP disclosed
US-5300643-A Viricides BAYER AKTIENGESELLSCHAFT (DE) 1994-04-05 US disclosed
US-5217972-A QUINOLONECARBOXYLIC ACID DERIVATIVES AND THEIR USE AS ANTIVIRAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1993-06-08 US disclosed
EP-0422485-A2 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1991-04-17 EP disclosed