Bicarbonate

Bicarbonate

SCHEMBL9044272

O=C(O)O.O=c1ccn(-c2ccc(F)cc2)c2cc(F)ccc12

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.47
KDM4E B2RXH2 5/20 0.43
LMNA P02545 4/20 0.43
KCNH2 Q12809 3/20 0.43
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 6/20 0.40
HPGD P15428 5/20 0.40
HSD17B10 Q99714 2/20 0.40
MAPT P10636 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
TSHR P16473 1/20 0.40
ALOX12 P18054 1/20 0.40
RAB9A P51151 1/20 0.40
CYP3A4 P08684 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL9044839 0.82 HTR1A (0.38) RORCLMNAKMT2ACYP2C9CYP3A4
Bicarbonate SCHEMBL9046002 0.80 MAPK8 (0.47) RORCKDM4EMAPTCYP2C9SMN1; SMN2
SCHEMBL9055849 0.75 MAOA (0.45) LMNAMAPT
SCHEMBL9044266 0.72 TDP1 (0.44) RORCKDM4ELMNAKMT2AALDH1A1
SCHEMBL1883370 0.71 KDM4E (0.45) RORCKDM4ELMNAKCNH2KMT2A
SCHEMBL31533281 0.70 ATM (0.40) LMNAALDH1A1MAPT
SCHEMBL10627492 0.70 ATM (0.47) KDM4EALDH1A1CYP2C9CYP2C19
SCHEMBL14984898 0.70 ALDH1A1 (0.41) RORCKDM4ELMNAKCNH2ALDH1A1
SCHEMBL1876893 0.70 LMNA (0.43) KDM4ELMNAKMT2AALDH1A1HPGD
SCHEMBL10475470 0.70 KCNH2 (0.58) RORCKDM4ELMNAKCNH2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422485-B1 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1996-04-03 EP disclosed
EP-0422485-A2 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1991-04-17 EP disclosed