Bicarbonate

Bicarbonate

SCHEMBL9044839

O=C(O)O.O=c1ccn(-c2ccc(F)cc2F)c2cc(F)ccc12

nearest known ligand 0.43

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B known ✓ P49841 1/20 0.38
HTR1A P08908 1/20 0.38
HTR2A P28223 1/20 0.38
HTR7 P34969 1/20 0.38
HTR6 P50406 1/20 0.38
RORC P51449 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CAPN1 P07384 1/20 0.38
EPHA2 P29317 1/20 0.38
FLT4 P35916 1/20 0.38
RARB P10826 1/20 0.38
TBXAS1 P24557 1/20 0.38
SLC6A3 Q01959 1/20 0.38
MAPK8 P45983 3/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
FFAR4 Q5NUL3 1/20 0.37
KMT2A Q03164 2/20 0.36
ATM Q13315 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL9046002 0.89 MAPK8 (0.47) RORCMAPK8CYP3A4CYP2C9ATM
SCHEMBL10593432 0.84 GLA (0.35) HTR1AHTR2AHTR7HTR6L3MBTL1
Bicarbonate SCHEMBL9044272 0.82 RORC (0.47) RORCCYP3A4CYP2C9KMT2AMEN1
SCHEMBL9147090 0.81 EPHA2 (0.53) RORCCAPN1EPHA2FLT4GSK3B
SCHEMBL9416468 0.76 MAPK8 (0.43) L3MBTL1CAPN1EPHA2FLT4GSK3B
Bicarbonate SCHEMBL9046548 0.74 PTGS1 (0.43) RORCMAPK8CYP3A4CYP2C9KMT2A
SCHEMBL500692 0.74 LMNA (0.56) CAPN1EPHA2FLT4GSK3BRARB
SCHEMBL9044837 0.73 GLA (0.40) L3MBTL1EPHA2FLT4GSK3BRARB
SCHEMBL2087613 0.73 LMNA (0.53) RORCEPHA2FLT4GSK3BRARB
SCHEMBL6216178 0.73 LMNA (0.50) HTR1AHTR2AHTR7HTR6RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422485-B1 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1996-04-03 EP disclosed
EP-0422485-A2 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1991-04-17 EP disclosed