SCHEMBL9047405

SCHEMBL9047405

Oc1n[c]nc2nc[nH]c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
PI4KA P42356 2/20 0.35
PI4K2B Q8TCG2 2/20 0.35
PI4K2A Q9BTU6 2/20 0.35
PI4KB Q9UBF8 2/20 0.35
LRRK2 Q5S007 2/20 0.35
LMNA P02545 1/20 0.35
DRD3 P35462 1/20 0.35
XDH P47989 1/20 0.35
PDPK1 O15530 3/20 0.34
GDA Q9Y2T3 1/20 0.34
G6PD P11413 1/20 0.34
CYP1A2 P05177 1/20 0.34
HIF1A Q16665 1/20 0.34
BRAF P15056 2/20 0.33
ADORA3 P0DMS8 2/20 0.33
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
CDK2 P24941 2/20 0.32
CHEK1 O14757 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8583607 0.75 PI4KA (0.53) ALDH1A1PI4KAPI4K2BPI4K2API4KB
SCHEMBL546075 0.71 XDH (0.53) ALDH1A1LMNAXDHCYP1A2HIF1A
SCHEMBL545952 0.71 PDPK1 (0.58) ALDH1A1PI4KAPI4K2BPI4K2API4KB
Hypoxanthine SCHEMBL25382 0.70 LMNA (0.57) ALDH1A1PI4KAPI4K2BPI4K2API4KB
SCHEMBL2346676 0.69 MKNK1 (0.41) ALDH1A1GDACYP1A2HIF1ABRAF
Xanthine SCHEMBL4966 0.68 GDA (0.44) ALDH1A1PI4KAPI4K2BPI4K2API4KB
Hypoxanthine SCHEMBL1230632 0.68 LMNA (0.55) ALDH1A1PI4KAPI4K2BPI4K2API4KB
SCHEMBL2696766 0.68 ALDH1A1 (0.41) ALDH1A1PI4KAPI4K2BPI4K2API4KB
Hypoxanthine SCHEMBL6673817 0.68 LMNA (0.55) ALDH1A1PI4KAPI4K2BPI4K2API4KB
Hypoxanthine SCHEMBL560393 0.68 PI4KA (0.59) ALDH1A1PI4KAPI4K2BPI4K2API4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0448726-B1 2-SUBSTITUTED 2-CYCLOPENTENONE AND CARCINOSTATIC AGENT AND OSTEOGENESIS PROMOTER CONTAINING THE SAME AS ACTIVE INGREDIENT TEIJIN LTD (JP) 1996-04-24 EP disclosed
US-5338844-A 2-substituted-2-cyclopentenone compound and anticancer agent and bone formation accelerator comprising same as active ingredient TEIJIN LIMITED (JP) 1994-08-16 US disclosed
US-5216183-A Antitumor, anticarcinogenic agents; bone formation accelerators TEIJIN LIMITED (JP) 1993-06-01 US disclosed
EP-0448726-A1 2-SUBSTITUTED 2-CYCLOPENTENONE AND CARCINOSTATIC AGENT AND OSTEOGENESIS PROMOTER CONTAINING THE SAME AS ACTIVE INGREDIENT TEIJIN LIMITED (JP) 1991-10-02 EP disclosed