SCHEMBL9047485

SCHEMBL9047485

COC1=Cc2cccc(OC)c2CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 1/20 0.41
DRD2 P14416 4/20 0.40
DRD3 P35462 4/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CHRM2 P08172 3/20 0.39
CHRM1 P11229 3/20 0.39
CHRM3 P20309 3/20 0.39
DRD1 P21728 1/20 0.39
DRD5 P21918 1/20 0.39
KDM4E B2RXH2 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5784077 0.79 ALDH1A1 (0.40) ALDH1A1CYP3A4DRD2DRD3CA12
SCHEMBL30715537 0.79 ALDH1A1 (0.40) ALDH1A1CYP3A4DRD2DRD3CA12
SCHEMBL22557831 0.77 DRD2 (0.41) ALDH1A1CYP3A4DRD2DRD3CA1
SCHEMBL29398439 0.77 DRD2 (0.41) ALDH1A1CYP3A4DRD2DRD3CA1
SCHEMBL22558013 0.77 PTGS2 (0.45) ALDH1A1CYP3A4DRD2DRD3CA12
SCHEMBL7777402 0.75 NOTUM (0.38) ALDH1A1CYP3A4DRD2DRD3CHRM2
SCHEMBL7779663 0.75 DRD2 (0.39) ALDH1A1CYP3A4DRD2DRD3CHRM2
SCHEMBL5780342 0.75 ENPP2 (0.43) ALDH1A1CYP3A4DRD2DRD3CHRM2
SCHEMBL9361584 0.75 DRD2 (0.38) ALDH1A1CYP3A4DRD2DRD3CHRM2
SCHEMBL7772436 0.74 SRD5A1 (0.51) ALDH1A1CYP3A4CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1035001-C Substituted phenyl phenol leukotriene antagonists LILLY CO ELI (US) 1997-05-28 CN disclosed
WO-1996036347-A1 USE OF LEUKOTRIENE ANTAGONISTS FOR ALZHEIMER'S DISEASE ELI LILLY AND COMPANY (US) 1996-11-21 WO disclosed
EP-0743064-A1 Leukotriene antagonists for use in the treatment or prevention of alzheimer's disease ELI LILLY AND COMPANY (US) 1996-11-20 EP disclosed
US-5462954-A Antiinflammatory, antiallergens; treating asthma ELI LILLY AND COMPANY (US) 1995-10-31 US disclosed
CN-1088906-A The phenyl phenol leukotriene antagonists that replaces LILLY CO ELI (US) 1994-07-06 CN disclosed
EP-0544488-A2 Substituted phenyl phenol leukotriene antagonists ELI LILLY AND COMPANY (US) 1993-06-02 EP disclosed