SCHEMBL9048832

SCHEMBL9048832

O=C(CCCl)c1cn(C(=O)CCCl)c2ccc(F)cc12

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.40
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
HTR3A P46098 10/20 0.35
RORC P51449 1/20 0.34
IDO1 P14902 1/20 0.34
HTR6 P50406 2/20 0.34
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9046975 0.81 AKR1C3 (0.44) AKR1C3AKR1C2HTR6
SCHEMBL9047869 0.80 KMT2A (0.50) HTR3A
SCHEMBL5790264 0.74 HTR6 (0.49) AKR1C3HTR6
SCHEMBL28436678 0.73 PTGDR2 (0.48) KCNH2HTR6
SCHEMBL6384689 0.70 HTR7 (0.50)
SCHEMBL959448 0.70 CES2 (0.57)
SCHEMBL27617465 0.69 AKR1C3 (0.40) KCNH2AKR1C3AKR1C2HTR6CNR2
SCHEMBL10768717 0.68 CHRNA7 (0.46)
SCHEMBL7278172 0.67 ALDH1A1 (0.46) KCNH2HTR6CNR2
SCHEMBL28436683 0.66 PTGDR2 (0.47) KCNH2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714896-A1 INDOL DERIVATIVES USEFUL FOR THE TREATMENT OF MIGRAINE, COMPOSITION AND UTILIZATION VITA-INVEST, S.A. (ES) 1996-06-05 EP disclosed