SCHEMBL904949

SCHEMBL904949

FC(F)(F)c1ccc(C(CCCN2CCC(N3CCc4ccccc43)CC2)c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.46
MTR Q99707 1/20 0.43
OPRM1 P35372 4/20 0.43
OPRL1 P41146 2/20 0.43
HTR1A P08908 6/20 0.43
OPRK1 P41145 3/20 0.43
SLC6A2 P23975 3/20 0.43
SLC6A4 P31645 3/20 0.43
DRD3 P35462 3/20 0.43
KCNH2 Q12809 3/20 0.43
OPRD1 P41143 2/20 0.43
CCR5 P51681 2/20 0.43
MEN1 O00255 2/20 0.43
CACNA1F O60840 2/20 0.43
GMNN O75496 2/20 0.43
USP2 O75604 2/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 2/20 0.43
CHRM2 P08172 2/20 0.43
ABCB1 P08183 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL904839 0.88 DRD3 (0.54) SIGMAR1MTROPRM1OPRL1HTR1A
SCHEMBL904928 0.83 SIGMAR1 (0.50) SIGMAR1MTROPRM1OPRL1HTR1A
SCHEMBL5870875 0.81 OPRM1 (0.43) SIGMAR1OPRM1OPRL1OPRK1DRD3
SCHEMBL14349454 0.79 OPRM1 (0.53) OPRM1OPRL1OPRK1DRD3KCNH2
SCHEMBL5871383 0.79 DRD3 (0.51) SIGMAR1DRD3CYP1A2DRD2HTR2A
SCHEMBL14282272 0.78 OPRM1 (0.52) OPRM1OPRL1OPRK1DRD3OPRD1
SCHEMBL3881201 0.74 OPRM1 (0.56) SIGMAR1OPRM1OPRL1HTR1AOPRK1
Fluorobenzene SCHEMBL27495584 0.73 DRD3 (0.47) SIGMAR1OPRM1OPRL1OPRK1DRD3
SCHEMBL904899 0.72 CCR3 (0.59) RAB9ANPSR1
SCHEMBL5871299 0.72 ACHE (0.54) SIGMAR1OPRM1OPRL1OPRK1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011143444-A2 DIPHENYLBUTYPIPERIDINE AUTOPHAGY INDUCERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2011-11-17 WO disclosed