SCHEMBL9050185

SCHEMBL9050185

Cc1nnc(NC(=O)C2CCc3nc[nH]c3C2)s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 6/20 0.45
HSD17B10 Q99714 3/20 0.44
HPGD P15428 2/20 0.44
HTR3A P46098 2/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
SLC6A4 P31645 1/20 0.43
OPRK1 P41145 1/20 0.43
HTR2B P41595 1/20 0.43
KCNH2 Q12809 1/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TP53 P04637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9050178 0.91 KMT2A (0.52) KMT2AMEN1KDM4EALDH1A1HSD17B10
SCHEMBL9049451 0.77 NPC1 (0.48) KMT2AMEN1ALDH1A1HSD17B10HPGD
SCHEMBL7327993 0.77 HTR3A (0.50) KDM4EALDH1A1HTR3AADRA2AADRA2B
SCHEMBL8542781 0.76 HTR3A (0.50) KDM4EHTR3AADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL9050935 0.76 HTR3A (0.48) ALDH1A1HTR3AADRA2AADRA2BADRA2C
SCHEMBL7333796 0.74 ADRA1A (0.47) KMT2AMEN1ALDH1A1HPGDHTR3A
SCHEMBL12648964 0.73 KMT2A (0.84) KMT2AMEN1KDM4EALDH1A1HSD17B10
SCHEMBL7328013 0.73 HTR3A (0.41) HTR3AADRA2AADRA2BADRA2CSLC6A4
SCHEMBL7324856 0.73 HTR3A (0.51) KDM4EALDH1A1HSD17B10HPGDHTR3A
SCHEMBL8482518 0.73 PDK1 (0.49) KMT2AKDM4EALDH1A1HTR3AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381422-B1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-10-23 EP disclosed
US-5496942-A 5-HT3-RECEPTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
US-5344927-A 5-HT3 antagonist YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-09-06 US disclosed
EP-0381422-A1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1990-08-08 EP disclosed