SCHEMBL9050178

SCHEMBL9050178

Cc1nnc(NC(=O)C2CCc3[nH]cnc3C2)s1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 6/20 0.45
HSD17B10 Q99714 3/20 0.44
HPGD P15428 3/20 0.44
TP53 P04637 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
PKM P14618 1/20 0.40
CHKA P35790 1/20 0.39
GAA P10253 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9050185 0.91 KMT2A (0.52) KMT2AMEN1KDM4EALDH1A1HSD17B10
SCHEMBL7327986 0.77 L3MBTL1 (0.47) KMT2AMEN1KDM4EALDH1A1TP53
SCHEMBL1417641 0.76 HTR3A (0.40) KDM4E
Hydrochloric Acid SCHEMBL9050917 0.76 HTR3A (0.39) ALDH1A1HPGDNPSR1LMNA
SCHEMBL6851321 0.76 HPGD (0.48) KMT2AMEN1KDM4EHSD17B10HPGD
SCHEMBL9049386 0.76 CYP1A2 (0.49) KMT2AMEN1KDM4EALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL6846874 0.75 HTR3A (0.39) KDM4E
SCHEMBL13531389 0.74 HTR3A (0.42) KDM4EALDH1A1SMN1; SMN2GAA
SCHEMBL13531413 0.74 HTR3A (0.42) KDM4EALDH1A1SMN1; SMN2GAA
SCHEMBL7333785 0.74 MMP8 (0.47) KMT2AMEN1ALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381422-B1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-10-23 EP disclosed
US-5496942-A 5-HT3-RECEPTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
US-5344927-A 5-HT3 antagonist YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-09-06 US disclosed
EP-0381422-A1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1990-08-08 EP disclosed