SCHEMBL9050587

SCHEMBL9050587

O=C1c2ccccc2OCN1CCN1CCN(c2ccccn2)CC1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 4/20 0.56
DRD1 P21728 3/20 0.56
DRD2 P14416 5/20 0.54
ADRA1D P25100 1/20 0.52
ADRA1A P35348 1/20 0.52
ADRA1B P35368 1/20 0.52
HTR1A P08908 5/20 0.50
HTR2A P28223 4/20 0.50
HTR7 P34969 4/20 0.50
HTR6 P50406 4/20 0.50
POLB P06746 1/20 0.48
KCNH2 Q12809 1/20 0.48
HTR2C P28335 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9049140 0.89 HTR1A (0.56) DRD3DRD1DRD2ADRA1DADRA1A
SCHEMBL9373187 0.83 DRD3 (0.68) DRD3DRD1DRD2HTR1AHTR2A
SCHEMBL9369214 0.83 DRD3 (0.68) DRD3DRD1DRD2HTR1AHTR2A
SCHEMBL9047511 0.83 HTR1A (0.54) DRD3DRD2ADRA1DADRA1AADRA1B
SCHEMBL6716162 0.80 DRD3 (0.69) DRD3DRD1DRD2ADRA1DADRA1A
SCHEMBL9049252 0.79 ADRA1B (0.57) ADRA1DADRA1AADRA1BHTR1AHTR7
SCHEMBL9372762 0.78 DRD3 (0.61) DRD3DRD1DRD2ADRA1DADRA1A
SCHEMBL13711971 0.78 KCNH2 (0.71) DRD3DRD1DRD2HTR1AHTR2A
SCHEMBL2518183 0.77 ADRA1D (0.71) DRD3DRD1DRD2ADRA1DADRA1A
SCHEMBL9048565 0.77 KCNH2 (0.53) DRD2HTR1AHTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0527081-B1 Substituted 3-piperazinylalkyl-2,3-dihydro-4H-1,3-benzoxazine-4-ones, their preparation and their therapeutical use PF MEDICAMENT (FR) 1996-01-03 EP claimed
US-5308844-A ANTIDEPRESSANT, ANXIOLYTIC AGENT, ANALGESIC, HYPOTENSIVE AGENT PIERRE FABRE MEDICAMENT (FR) 1994-05-03 US disclosed