SCHEMBL9053391

SCHEMBL9053391

CN1CCc2ccc(-c3cn(-c4ccc(CCC(=O)O)cc4)cn3)cc2CC1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DVL1 O14640 1/20 0.44
RXRA P19793 2/20 0.42
RXRB P28702 2/20 0.42
RXRG P48443 2/20 0.42
ESR1 P03372 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
FFAR4 Q5NUL3 6/20 0.39
MAP4K4 O95819 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
FFAR1 O14842 2/20 0.37
TBXAS1 P24557 2/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9056558 0.88 RXRA (0.42) DVL1RXRARXRBRXRGFFAR4
SCHEMBL9057943 0.81 DVL1 (0.50) DVL1RXRARXRBRXRGESR1
SCHEMBL9054062 0.80 MELK (0.41) DVL1RXRARXRBRXRGESR1
Hydrochloric Acid SCHEMBL9062779 0.80 DVL1 (0.49) DVL1RXRARXRBRXRGESR1
Hydrochloric Acid SCHEMBL9057996 0.78 DVL1 (0.45) DVL1RXRARXRBRXRGESR1
Hydrochloric Acid SCHEMBL9057948 0.78 DVL1 (0.56) DVL1RXRARXRBRXRGPIM2
SCHEMBL9055061 0.78 S1PR1 (0.48) DVL1RXRARXRBRXRGHRH3
SCHEMBL9255613 0.75 ITGB3 (0.58) RXRARXRBRXRGMAP4K4FFAR1
SCHEMBL8559863 0.74 S1PR1 (0.50) RXRARXRBRXRGESR1HRH3
Hydrochloric Acid SCHEMBL8563445 0.73 S1PR1 (0.49) RXRARXRBRXRGESR1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004271-A1 CONDENSED AZEPINE DERIVATIVES, DRUGS CONTAINING THESE COMPOUNDS AND METHODS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-02-15 WO disclosed