SCHEMBL9055252

SCHEMBL9055252

CC(Nc1ccc([N+](=O)[O-])c2c(C#N)cccc12)c1ccncc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.42
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
LRRK2 Q5S007 1/20 0.38
ALDH1A1 P00352 6/20 0.38
HPGD P15428 3/20 0.38
MAPT P10636 5/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
HTR6 P50406 1/20 0.36
CTSB P07858 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
TP53 P04637 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9056096 0.89 CRHBP (0.37) POLBCRHBPCRHR2ALDH1A1HPGD
SCHEMBL9054862 0.83 POLB (0.40) POLBCRHBPCRHR2LRRK2ALDH1A1
SCHEMBL9055492 0.74 HTT (0.54) POLBALDH1A1HPGDMAPTKDM4E
SCHEMBL9055262 0.70 TYMS (0.47) POLBLRRK2ALDH1A1MAPTMAPK1
SCHEMBL9055272 0.69 CTSB (0.40) ALDH1A1MAPTCTSBMEN1KMT2A
SCHEMBL11811062 0.69 TDP1 (0.55) POLBALDH1A1HPGDMAPTGAA
SCHEMBL9055280 0.69 ALDH1A1 (0.47) ALDH1A1MAPTMAPK1KDM4EGAA
SCHEMBL9055020 0.69 TDP1 (0.42) POLBALDH1A1MAPTSMN1; SMN2GAA
SCHEMBL16756262 0.65 MAPT (0.59) POLBCRHBPCRHR2ALDH1A1HPGD
SCHEMBL16756260 0.65 MAPT (0.59) POLBCRHBPCRHR2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545744-A Cyano naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-08-13 US disclosed
US-5498727-A Preparation of benzindole compounds from naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-03-12 US disclosed
WO-1996002502-A1 PREPARATION OF BENZINDOLE COMPOUNDS FROM NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1996-02-01 WO disclosed