SCHEMBL9055513

SCHEMBL9055513

O=C1Nc2c(cc(S(=O)(=O)N3CCCC3)c3c2CCCC3)C1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.47
CASP1 P29466 2/20 0.47
CASP7 P55210 2/20 0.47
CASP9 P55211 1/20 0.47
ALDH1A1 P00352 7/20 0.40
TSHR P16473 3/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
POLB P06746 2/20 0.39
USP2 O75604 1/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CES1 P23141 1/20 0.38
DNMT1 P26358 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9057244 0.99 CASP3 (0.48) CASP3CASP1CASP7CASP9ALDH1A1
SCHEMBL9055289 0.86 ALDH1A1 (0.42) CASP3CASP1CASP7CASP9ALDH1A1
SCHEMBL9207029 0.82 CES1 (0.40) CASP3CASP1CASP7CASP9ALDH1A1
SCHEMBL9055477 0.82 CES1 (0.41) CASP3CASP1CASP7CASP9ALDH1A1
SCHEMBL9056121 0.78 CES1 (0.39) CASP3ALDH1A1TSHRCYP3A4CYP2C9
SCHEMBL9056485 0.75 TSHR (0.38) CASP1CASP7ALDH1A1TSHRCYP3A4
SCHEMBL23412593 0.73 ALDH1A1 (0.49) ALDH1A1CES1DNMT1
SCHEMBL23412305 0.70 ALDH1A1 (0.49) ALDH1A1CES1DNMT1
Hydrochloric Acid SCHEMBL8326999 0.69 ALDH1A1 (0.39) CASP3CASP1CASP7CASP9ALDH1A1
Hydrochloric Acid SCHEMBL8326997 0.69 ALDH1A1 (0.39) CASP3CASP1CASP7CASP9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0522494-B1 Novel isatineoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1996-10-02 EP disclosed
US-5223527-A Isatineoxime derivatives and their use NEUROSEARCH A/S (DK) 1993-06-29 US disclosed
EP-0522494-A1 Novel isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-01-13 EP disclosed