SCHEMBL9057934

SCHEMBL9057934

CSc1cc(C)nc(SC)c1NC(=O)N(Cc1ccc(Oc2ccc(F)cc2)cc1)C1CCOCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
HTR2A P28223 11/20 0.38
SCN9A Q15858 1/20 0.38
ABCB11 O95342 1/20 0.37
CYP1A2 P05177 1/20 0.37
ADRB2 P07550 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
DRD1 P21728 1/20 0.37
TBXA2R P21731 1/20 0.37
SLC6A2 P23975 1/20 0.37
HTR2C P28335 1/20 0.37
GPR183 P32249 1/20 0.37
CYP2C19 P33261 1/20 0.37
ADRA1A P35348 1/20 0.37
OPRM1 P35372 1/20 0.37
APLNR P35414 1/20 0.37
DRD3 P35462 1/20 0.37
CX3CR1 P49238 1/20 0.37
SLC6A3 Q01959 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8807728 0.92 TP53 (0.42) TP53HTR2ASCN9AABCB11CYP1A2
SCHEMBL8809049 0.92 TP53 (0.42) TP53HTR2ASCN9AABCB11CYP1A2
SCHEMBL29972806 0.92 TP53 (0.42) TP53HTR2ASCN9AABCB11CYP1A2
SCHEMBL8807796 0.85 THRB (0.39) TP53CYP1A2CYP2C19UBE2MDCUN1D1
SCHEMBL8808860 0.84 USP2 (0.43) TP53CYP1A2CYP2C19UBE2MDCUN1D1
SCHEMBL9056629 0.83 KMT2A (0.38) TP53CYP1A2CYP2C19UBE2MDCUN1D1
SCHEMBL9058046 0.83 UBE2M (0.41) HTR2ACYP1A2CYP2C19UBE2MDCUN1D1
SCHEMBL8808573 0.83 LPAR1 (0.41) TP53CYP1A2CYP2C19
SCHEMBL9059535 0.83 TP53 (0.41) TP53HTR2AABCB11CYP1A2ADRB2
SCHEMBL8808548 0.83 TP53 (0.41) TP53HTR2AABCB11CYP1A2ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996010559-A1 UREA DERIVATIVES AND THEIR USE AS ACAT-INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-04-11 WO disclosed