SCHEMBL9064941

SCHEMBL9064941

CC(=O)c1ccc(N2C(=O)C=C(C)C2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.46
ADAM17 P78536 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.41
TSHR P16473 1/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
DDAH1 O94760 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HTT P42858 1/20 0.41
CACNA1B Q00975 1/20 0.41
APBA1 Q02410 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 1/20 0.40
KCNJ1 P48048 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CA9 Q16790 4/20 0.39
CA12 O43570 3/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8442000 0.86 DDAH1 (0.58) KMT2AL3MBTL1ALDH1A1HPGDDDAH1
SCHEMBL94147 0.85 MGLL (0.46) KMT2AHSP90AA1NPSR1TDP1MEN1
SCHEMBL11251677 0.85 CA9 (0.39) KMT2AALDH1A1HPGDDDAH1HSP90AA1
SCHEMBL22152298 0.83 NSD2 (0.41) KMT2ATSHRHSP90AA1TDP1MEN1
SCHEMBL22601779 0.82 MEN1 (0.38) KMT2ATSHRALDH1A1HPGDDDAH1
SCHEMBL14579489 0.81 PARP1 (0.51) KMT2AL3MBTL1TSHRALDH1A1HSP90AA1
SCHEMBL8443563 0.80 MGLL (0.53) KMT2AALDH1A1HSP90AA1HTTNPSR1
SCHEMBL13477928 0.80 KMT2A (0.50) KMT2AALDH1A1HPGDHSP90AA1HTT
SCHEMBL13477929 0.80 RAB9A (0.51) KMT2AL3MBTL1ALDH1A1HPGDHSP90AA1
SCHEMBL8142750 0.80 MGLL (0.57) KMT2ATSHRALDH1A1CACNA1BAPBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110235292-A1 THERMOSETTING COMPOSITION AND PRINTED CIRCUIT BOARD USING THE SAME SAMSUNG ELECTRONICS CO., LTD. (KR) 2011-09-29 US disclosed
US-20110235292-A1 THERMOSETTING COMPOSITION AND PRINTED CIRCUIT BOARD USING THE SAME SAMSUNG ELECTRONICS CO., LTD. (KR) 2011-09-29 US disclosed
US-5523360-A IMPROVES MELT-FLOW PROPERTIES AKZO NOBEL N. V. (NL) 1996-06-04 US disclosed
EP-0648240-A1 PROCESS FOR THE MODIFICATION OF POLYPHENYLENE ETHER RESIN COMPOSITIONS Akzo Nobel N.V. (NL) 1995-04-19 EP disclosed
EP-0495545-B1 Citraconimide (co)polymers and curing with anionic catalyst AKZO NOBEL NV (NL) 1994-12-28 EP disclosed
WO-1994001485-A1 PROCESS FOR THE MODIFICATION OF POLYPHENYLENE ETHER RESIN COMPOSITIONS AKZO NOBEL N.V. (NL) 1994-01-20 WO disclosed
US-5221717-A CITRACONIMIDE (CO)POLYMERS AND CURING WITH ANIONIC CATALYST AKZO N.V. (NL) 1993-06-22 US disclosed
EP-0495545-A1 Citraconimide (co)polymers and curing with anionic catalyst Akzo Nobel N.V. (NL) 1992-07-22 EP disclosed