SCHEMBL8443563

SCHEMBL8443563

CC1=CC(=O)N(c2ccc(O)cc2)C1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 3/20 0.53
HSP90AA1 P07900 1/20 0.53
PKM P14618 1/20 0.53
MAPK1 P28482 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
APAF1 O14727 1/20 0.48
POLB P06746 1/20 0.48
ESR1 P03372 5/20 0.46
ESR2 Q92731 3/20 0.46
KMT2A Q03164 4/20 0.44
NR1H3 Q13133 1/20 0.41
MEN1 O00255 3/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
F2 P00734 1/20 0.38
ELANE P08246 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL94147 0.90 MGLL (0.46) MGLLHSP90AA1PKMMAPK1NPSR1
SCHEMBL8142750 0.84 MGLL (0.57) MGLLMAPK1KMT2AMEN1ALDH1A1
SCHEMBL4839640 0.82 MGLL (0.61) MGLLHSP90AA1PKMMAPK1NPSR1
SCHEMBL8884854 0.81 CCR6 (0.35) MGLLHSP90AA1PKMMAPK1NPSR1
SCHEMBL9065005 0.81 MGLL (0.53) MGLLHSP90AA1MAPK1NPSR1POLB
SCHEMBL28434063 0.81 MGLL (0.53) MGLLPOLBKMT2AMEN1KDM4E
SCHEMBL26659413 0.81 ALDH1A1 (0.46) MGLLMAPK1NPSR1ESR2KMT2A
SCHEMBL10704906 0.81 MEN1 (0.56) MGLLNPSR1POLBKMT2AMEN1
SCHEMBL8442000 0.80 DDAH1 (0.58) NPSR1TDP1POLBKMT2AMEN1
SCHEMBL9064941 0.80 KMT2A (0.46) HSP90AA1NPSR1TDP1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111316986-B Application of maleimide compound as chitin synthetase inhibitor 浙江工业大学 2021-10-15 CN disclosed
CN-111316986-A Application of maleimide compound as chitin synthetase inhibitor 浙江工业大学 2020-06-23 CN disclosed
CN-107162950-A N substitution maleimide compounds and its preparation based on pharmaceutical intermediate are studied with antibacterial activity 浙江工业大学 2017-09-15 CN disclosed
EP-0495544-B1 Process for the synthesis of citraconimides AKZO NOBEL NV (NL) 1999-04-07 EP disclosed
US-5523360-A IMPROVES MELT-FLOW PROPERTIES AKZO NOBEL N. V. (NL) 1996-06-04 US disclosed
EP-0648240-A1 PROCESS FOR THE MODIFICATION OF POLYPHENYLENE ETHER RESIN COMPOSITIONS Akzo Nobel N.V. (NL) 1995-04-19 EP disclosed
EP-0495545-B1 Citraconimide (co)polymers and curing with anionic catalyst AKZO NOBEL NV (NL) 1994-12-28 EP disclosed
WO-1994001485-A1 PROCESS FOR THE MODIFICATION OF POLYPHENYLENE ETHER RESIN COMPOSITIONS AKZO NOBEL N.V. (NL) 1994-01-20 WO disclosed
US-5221717-A CITRACONIMIDE (CO)POLYMERS AND CURING WITH ANIONIC CATALYST AKZO N.V. (NL) 1993-06-22 US disclosed
EP-0495545-A1 Citraconimide (co)polymers and curing with anionic catalyst Akzo Nobel N.V. (NL) 1992-07-22 EP disclosed