SCHEMBL9080432

SCHEMBL9080432

CC(C)(C)c1ccc2c(CO[SiH](c3ccccc3)c3ccccc3)c(CBr)ccc2c1

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.32
CYP2D6 P10635 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KIF11 P52732 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701313 0.88 CYP2D6 (0.35) NR1I2CYP2D6ALDH1A1CYP1A2CYP2C19
SCHEMBL8849619 0.73 CYP2D6 (0.38) CYP2D6ALDH1A1CYP1A2CYP2C19
SCHEMBL8055340 0.72 CYP2D6 (0.40) CYP2D6ALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL9704031 0.71 KIF11 (0.31) KIF11
SCHEMBL9347229 0.70 CYP2D6 (0.54) CYP2D6ALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL9080434 0.70 NR1I2 (0.32) NR1I2CYP2D6KIF11
SCHEMBL9347249 0.69 CYP2D6 (0.37) CYP2D6ALDH1A1
SCHEMBL1206899 0.68 NR1I2 (0.32) NR1I2
SCHEMBL9472706 0.68 CYP2D6 (0.33) CYP2D6ALDH1A1
SCHEMBL9472693 0.67 GPR84 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5574039-A ANTITUMOR, FUNGICIDES AGOURON PHARMACEUTICALS, INC. (US) 1996-11-12 US disclosed
EP-0550566-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS (US) 1993-07-14 EP disclosed
WO-1992005153-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1992-04-02 WO disclosed