SCHEMBL9092

SCHEMBL9092

Nc1cccc(Br)c1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.45
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
CA14 Q9ULX7 2/20 0.43
PRNP P04156 1/20 0.42
KDM4E B2RXH2 4/20 0.39
GLA P06280 1/20 0.39
MAPT P10636 3/20 0.36
G6PD P11413 1/20 0.36
CASP7 P55210 1/20 0.36
CASP6 P55212 1/20 0.36
GAA P10253 1/20 0.36
TDP1 Q9NUW8 2/20 0.35
MEN1 O00255 1/20 0.35
KDM6B O15054 1/20 0.35
KDM4A O75164 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzoic Acid SCHEMBL25345242 0.91 TSHR (0.50) MMP2CA12CA1CA2CA9
SCHEMBL11857403 0.86 MAPT (0.55) GLAMAPTGAATDP1MEN1
SCHEMBL1000014 0.84 MMP2 (0.54) MMP2CA12CA1CA2CA7
SCHEMBL570378 0.84 CA12 (0.52) CA12CA1CA2CA7CA9
SCHEMBL1502516 0.83 PARP1 (0.41) MMP2KDM4EMAPTGAATDP1
SCHEMBL1189236 0.81 THRB (0.45) MMP2KDM4EMAPTTDP1ALDH1A1
SCHEMBL19972022 0.81 ALDH1A1 (0.45) MMP2KDM4EMAPTCASP7GAA
SCHEMBL18043789 0.79 MMP2 (0.50) MMP2CA12CA1CA2CA7
SCHEMBL1189541 0.76 CA1 (0.52) CA12CA1CA2CA7CA9
SCHEMBL15520067 0.76 HDAC8 (0.42) CA2KDM4EGAAALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 366 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117659069-A Synthesis method of 2-methyl-5- (4, 5-tetramethyl-1, 3, 2-dioxaborolan-2-yl) quinoline 南通敏言生物医药科技有限公司 2024-03-08 CN claimed
CN-115010671-B One-step synthesis method of 2-substituted quinazolinone 江苏大学 2023-10-10 CN claimed
CN-115010671-A One-step synthesis method of 2-substituted quinazolinone 江苏大学 2022-09-06 CN claimed
CN-106995438-B A kind of substituted quinazoline -4- ketone compounds and preparation method thereof and medical usage 中国科学院上海药物研究所 2019-09-20 CN claimed
CN-106995438-A One class substituted quinazoline -4- ketone compounds and preparation method thereof and medical usage 中国科学院上海药物研究所 2017-08-01 CN claimed
US-4673740-A Preparation of substituted 2-phenyl-4H-3,1-benzoxazin-4-ones BASF AKTIENGESELLSCHAFT (DE) 1987-06-16 US claimed
CN-122036604-A Compound and application thereof 中国药科大学 2026-05-15 CN disclosed
EP-4695250-A1 TETRACYCLIC COMPOUNDS AS SMARCA2 AND/OR SMARCA4 DEGRADERS Aurigene Oncology Limited (IN) 2026-02-18 EP disclosed
EP-4680612-A1 CHEMICAL COMPOUNDS AN2 Therapeutics, Inc. (US) 2026-01-21 EP disclosed
US-20250361236-A9 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS GILEAD SCIENCES INC (US) 2025-11-27 US disclosed
US-20250230144-A1 QUINAZOLINES AS POTASSIUM ION CHANNEL INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2025-07-17 US disclosed
CN-120058621-A 2, 3-Dihydro quinazoline derivative containing substituted phenyl, preparation method and application thereof 中国医学科学院药物研究所 2025-05-30 CN disclosed
US-20240425475-A1 COMPOUND BASED ON QUINAZOLINE-SUBSTITUTED GLUTARIMIDE SKELETON AND USE THEREOF GLUETACS THERAPEUTICS (SHANGHAI) CO., LTD. (CN) 2024-12-26 US disclosed
EP-1717230-A1 FUSED-RING 4-OXOPYRIMIDINE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2006-11-02 EP disclosed
US-20050182045-A1 Fused ring 4-oxopyrimidine derivative BANYU PHARMACEUTICAL CO., LTD. (JP) 2005-08-18 US disclosed
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO disclosed
US-4673740-A Preparation of substituted 2-phenyl-4H-3,1-benzoxazin-4-ones BASF AKTIENGESELLSCHAFT (DE) 1987-06-16 US disclosed
US-4337270-A ANTIALLERGENS; ANTIANAPHYLACTIC AGENTS HISAMITSU PHARMACEUTICAL CO., INC. (JP) 1982-06-29 US disclosed
US-4154745-A Isobenzofuran route to anthracycloquinones RESEARCH CORPORATION (US) 1979-05-15 US disclosed
US-4116981-A 5,12-EPOXY-NAPHTHACENE-6,11-DIONE DERIVATIVES Tsay, Yuh-Geng (TW) 1978-09-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250230144-A1 QUINAZOLINES AS POTASSIUM ION CHANNEL INHIBITORS KCNJ4, KCNK4, KCNQ4 MMP2 4262/4885CA12 4859/4885CA1 4239/4885
US-20240425475-A1 COMPOUND BASED ON QUINAZOLINE-SUBSTITUTED GLUTARIMIDE SKELETON AND USE THEREOF CRBN, CLN6, CDR2 MMP2 3512/4885CA12 1261/4885CA1 292/4885
US-20050182045-A1 Fused ring 4-oxopyrimidine derivative HRH4, HRH2, HRH3 MMP2 4362/4885CA12 4020/4885CA1 2445/4885
US-20250361236-A9 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS DGKG, DGKB, DGKK MMP2 3159/4885CA12 4736/4885CA1 4831/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.