SCHEMBL9105786

SCHEMBL9105786

C#CCNC(=O)CC1C(=O)N(C(Cl)Cc2ccc(Cl)cc2)CC(=O)N1CC#C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.33
ITGB2 P05107 2/20 0.33
ICAM1 P05362 2/20 0.33
ITGAL P20701 2/20 0.33
MAPT P10636 3/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ALDH1A1 P00352 4/20 0.32
KDM4E B2RXH2 2/20 0.32
LMNA P02545 3/20 0.32
TSHR P16473 1/20 0.32
POLB P06746 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
BRD4 O60885 1/20 0.31
TP53 P04637 1/20 0.31
SDCBP O00560 1/20 0.31
SDC2 P34741 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9104473 0.92 LMNA (0.39) GPBAR1ITGB2ICAM1ITGALMAPT
SCHEMBL9105245 0.91 ALDH1A1 (0.41) MAPTALDH1A1KDM4ELMNATSHR
SCHEMBL3701796 0.89 MEN1 (0.35) MAPTHDAC1HDAC8HDAC6NPC1
SCHEMBL3701709 0.89 HPGD (0.40) GPBAR1MAPTHDAC1HDAC8HDAC6
SCHEMBL9099926 0.89 HDAC1 (0.32) GPBAR1ITGB2ICAM1ITGALMAPT
SCHEMBL9105229 0.89 ITGB2 (0.39) ITGB2ICAM1ITGALMAPTHDAC1
SCHEMBL9104212 0.88 ALDH1A1 (0.40) MAPTALDH1A1KDM4ELMNAPOLB
SCHEMBL3702422 0.88 GPBAR1 (0.35) GPBAR1ITGB2ICAM1ITGALHDAC1
SCHEMBL9107195 0.86 MEN1 (0.41) MAPTNPC1RAB9AALDH1A1TSHR
SCHEMBL3702498 0.86 HPGD (0.39) MAPTHDAC8ALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460798-A2 APAF-1 INHIBITOR COMPOUNDS Laboratorios SALVAT, S.A. (ES) 2012-06-06 EP disclosed