SCHEMBL9110239

SCHEMBL9110239

O=c1ccccn1-c1cccnc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.55
EP300 Q09472 1/20 0.51
KAT2B Q92831 1/20 0.51
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA9 Q16790 1/20 0.51
CA14 Q9ULX7 1/20 0.51
CYP2A6 P11509 3/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2E1 P05181 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.47
F10 P00742 1/20 0.47
CYP11B2 P19099 1/20 0.46
ELANE P08246 1/20 0.45
GAA P10253 2/20 0.44
MAPT P10636 2/20 0.44
HSD17B10 Q99714 2/20 0.44
MAPK1 P28482 1/20 0.44
AR P10275 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30080798 1.00 HTT (0.55) HTTEP300KAT2BCA12CA1
Hydrochloric Acid SCHEMBL30385194 0.98 HTT (0.53) HTTEP300KAT2BCA12CA1
SCHEMBL31063913 0.83 CA12 (0.41) HTTEP300KAT2BCA12CA1
SCHEMBL31134347 0.83 CYP2A6 (0.50) HTTEP300KAT2BCA12CA1
SCHEMBL31134309 0.83 CA12 (0.41) HTTEP300KAT2BCA12CA1
SCHEMBL3561936 0.79 CA12 (0.50) EP300KAT2BCA12CA1CA2
SCHEMBL143175 0.78 ALDH1A1 (0.54) EP300KAT2BF10GAAMAPT
SCHEMBL1044182 0.76 ELANE (0.45) CA12CA1CA2CA9CA14
SCHEMBL31310093 0.76 CYP2A6 (0.46) HTTEP300KAT2BCYP2A6CYP3A4
SCHEMBL27990226 0.76 CA12 (0.48) EP300KAT2BCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3768671-B1 SUBSTITUTED IMIDAZOLIDIN-2-ONE DERIVATIVES AS PRMT5 INHIBITORS AURIGENE ONCOLOGY LTD (IN) 2024-05-22 EP claimed
US-11542275-B2 Substituted imidazolidin-2-one derivatives as PRMT5 inhibitors AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2023-01-03 US claimed
EP-0127756-A1 Process for the preparation of 5-pyridyl-pyridine-2(1H)-ones FABRICA DE PRODUCTOS QUIMICOS Y FARMACEUTICOS ABELLO, S.A. (ES) 1984-12-12 EP claimed
CN-122079879-A Nitrogen-containing heterocyclic derivative inhibitor, preparation method and application thereof 2026-05-26 CN disclosed
CN-122079878-A Nitrogen-containing heterocyclic derivative inhibitor, preparation method and application thereof 2026-05-26 CN disclosed
CN-122079880-A Nitrogen-containing heterocyclic derivative inhibitor, preparation method and application thereof 2026-05-26 CN disclosed
CN-120476110-B Nitrogen-containing heterocyclic derivative inhibitor, preparation method and application thereof SHANGHAI HANSOH BIOMEDICAL Co.,Ltd. (CN) 2026-05-26 CN disclosed
US-20260085045-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI HANSOH BIOMEDICAL CO LTD (CN) 2026-03-26 US disclosed
US-12497366-B2 Nitrogen-containing heterocyclic derivative inhibitor, preparation method therefor and use thereof SHANGHAI HANSOH BIOMEDICAL CO., LTD. (CN) 2025-12-16 US disclosed
US-20250326722-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI HANSOH BIOMEDICAL CO LTD (CN) 2025-10-23 US disclosed
EP-4590396-A1 PCSK9 INHIBITORS AND METHODS OF USE THEREOF Astrazeneca AB (SE) 2025-07-30 EP disclosed
WO-2014074660-A1 ALKYL-AMIDE-SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AND/OR IFNα RESPONSES BRISTOL-MYERS SQUIBB COMPANY (US) 2014-05-15 WO disclosed
EP-2648516-A1 SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS Confluence Life Sciences, Inc. (US) 2013-10-16 EP disclosed
WO-2012078684-A1 SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS CONFLUENCE LIFE SCIENCES, INC. (US) 2012-06-14 WO disclosed
US-20120142709-A1 SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS ACLARIS THERAPEUTICS, INC. 2012-06-07 US disclosed
EP-0127756-B1 PROCESS FOR THE PREPARATION OF 5-PYRIDYL-PYRIDINE-2(1H)-ONES FABRICA DE PRODUCTOS QUIMICOS Y FARMACEUTICOS ABELLO, S.A. (ES) 1988-10-26 EP disclosed
US-4563528-A Process for preparing 5 pyridyl pyridine-2 (1H)-ones FABRICA DE PRODUCTOS QUIMICOS Y FARMACEUTICOS ABELLO, S.A. (ES) 1986-01-07 US disclosed
EP-0127756-A1 Process for the preparation of 5-pyridyl-pyridine-2(1H)-ones FABRICA DE PRODUCTOS QUIMICOS Y FARMACEUTICOS ABELLO, S.A. (ES) 1984-12-12 EP disclosed
EP-0127756-A1 Process for the preparation of 5-pyridyl-pyridine-2(1H)-ones FABRICA DE PRODUCTOS QUIMICOS Y FARMACEUTICOS ABELLO, S.A. (ES) 1984-12-12 EP disclosed
EP-0127756-A1 Process for the preparation of 5-pyridyl-pyridine-2(1H)-ones FABRICA DE PRODUCTOS QUIMICOS Y FARMACEUTICOS ABELLO, S.A. (ES) 1984-12-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11542275-B2 Substituted imidazolidin-2-one derivatives as PRMT5 inhibitors PRMT5, PRMT1, PRMT8 HTT 3608/4885EP300 868/4885KAT2B 1378/4885
US-20120142709-A1 SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS MAPK1, MAP3K1, MAP3K6 HTT 4247/4885EP300 1152/4885KAT2B 2688/4885
US-20260085045-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF NPR1, CBR1, NAT1 HTT 1422/4885EP300 2725/4885KAT2B 1466/4885
US-12497366-B2 Nitrogen-containing heterocyclic derivative inhibitor, preparation method therefor and use thereof WEE1, WEE2, NOS1 HTT 1356/4885EP300 3523/4885KAT2B 3687/4885
US-20250326722-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF WEE1, WEE2, NOS1 HTT 1356/4885EP300 3523/4885KAT2B 3687/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.